SCHEMBL15428428

SCHEMBL15428428

Fc1ccc(Nc2ncnc3ccsc23)c(OC2CCCC2)c1

nearest known ligand 0.63

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MKNK2 Q9HBH9 16/20 0.63
MKNK1 Q9BUB5 9/20 0.63
EIF4E P06730 2/20 0.63
AURKA O14965 1/20 0.43
TEK Q02763 1/20 0.43
AURKB Q96GD4 1/20 0.43
DYRK1A Q13627 1/20 0.41
DYRK1B Q9Y463 1/20 0.41
FADS1 O60427 1/20 0.41
EGFR P00533 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13434850 0.87 MKNK2 (0.59) MKNK2MKNK1EIF4EEGFR
SCHEMBL13434851 0.84 DYRK1A (0.55) MKNK2MKNK1EIF4EAURKATEK
SCHEMBL3803642 0.83 MKNK1 (0.57) MKNK2MKNK1EIF4EEGFR
SCHEMBL13434842 0.83 MKNK2 (0.44) MKNK2MKNK1EIF4EAURKAAURKB
SCHEMBL13434854 0.80 EGFR (0.47) MKNK2MKNK1EIF4EAURKATEK
SCHEMBL13434849 0.79 MKNK2 (0.53) MKNK2MKNK1EIF4EAURKATEK
SCHEMBL18839802 0.77 MKNK2 (0.61) MKNK2MKNK1EIF4E
SCHEMBL20575252 0.77 MKNK2 (1.00) MKNK2MKNK1EIF4E
SCHEMBL13434847 0.77 MKNK2 (0.54) MKNK2MKNK1EIF4EAURKATEK
SCHEMBL23049793 0.76 MKNK2 (0.98) MKNK2MKNK1EIF4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8633201-B2 Thienopyrimidines having Mnk1/Mnk2 inhibiting activity for pharmaceutical compositions BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-01-21 US disclosed