SCHEMBL15428772

SCHEMBL15428772

CN(C(=O)O)[C@H]1CC[C@H](Cn2ncc3cnc(Nc4ccc(C5CCCCC5)cc4)nc32)CC1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
AURKA O14965 12/20 0.44
CDK1 P06493 12/20 0.44
CCNB1 P14635 12/20 0.44
CDK4 P11802 3/20 0.42
CCND1 P24385 3/20 0.42
CCND2 P30279 1/20 0.42
CCND3 P30281 1/20 0.42
BRD4 O60885 1/20 0.41
CREBBP Q92793 1/20 0.41
DGAT1 O75907 1/20 0.39
JAK3 P52333 2/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
JAK1 P23458 1/20 0.39
LCK P06239 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL343335 0.86 AURKA (0.43) AURKACDK1CCNB1CDK4CCND1
SCHEMBL15428771 0.85 CDK4 (0.44) AURKACDK1CCNB1CDK4CCND1
SCHEMBL343810 0.83 CDK4 (0.49) AURKACDK1CCNB1CDK4CCND1
SCHEMBL15428739 0.83 JAK1 (0.44) AURKAJAK3JAK1
SCHEMBL343483 0.83 AURKA (0.46) AURKACDK1CCNB1CDK4CCND1
SCHEMBL343484 0.83 AURKA (0.46) AURKACDK1CCNB1CDK4CCND1
SCHEMBL343334 0.81 AURKA (0.41) AURKACDK1CCNB1CDK4CCND1
SCHEMBL15428702 0.80 CDK1 (0.41) AURKACDK1CCNB1CDK4CCND1
SCHEMBL15428749 0.80 JAK1 (0.47) JAK3JAK1
SCHEMBL15428718 0.79 CDK2 (0.47) AURKACDK1CCNB1CCND3JAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8637529-B2 Pyrazolo[3,4-d]pyrimidine compounds AbbYie Inc. (US) 2014-01-28 US disclosed