SCHEMBL1542883

SCHEMBL1542883

C[C@@H](CO)NC(=O)[C@@H]1CCC(NC(=O)c2ccc(-c3cccc(F)c3)nc2)C1

nearest known ligand 0.56

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HPGDS O60760 5/20 0.56
GABRA5 P31644 4/20 0.46
NPR1 P16066 2/20 0.45
CYP2C9 P11712 5/20 0.44
MAPK14 Q16539 5/20 0.44
MAPK11 Q15759 1/20 0.43
MAP4K4 O95819 1/20 0.43
WNT3A P56704 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13240650 1.00 HPGDS (0.56) HPGDSGABRA5NPR1CYP2C9MAPK14
SCHEMBL1542884 1.00 HPGDS (0.56) HPGDSGABRA5NPR1CYP2C9MAPK14
SCHEMBL3089298 0.95 HPGDS (0.54) HPGDSGABRA5NPR1CYP2C9MAPK14
SCHEMBL3088895 0.95 HPGDS (0.54) HPGDSGABRA5NPR1CYP2C9MAPK14
SCHEMBL3088898 0.95 HPGDS (0.54) HPGDSGABRA5NPR1CYP2C9MAPK14
SCHEMBL13572477 0.95 HPGDS (0.54) HPGDSGABRA5NPR1CYP2C9MAPK14
SCHEMBL3088900 0.95 HPGDS (0.54) HPGDSGABRA5NPR1CYP2C9MAPK14
SCHEMBL2988675 0.86 HPGDS (0.64) HPGDSGABRA5CYP2C9MAPK14MAPK11
SCHEMBL2996963 0.83 HPGDS (0.57) HPGDSGABRA5CYP2C9MAPK14MAPK11
SCHEMBL2986340 0.83 HPGDS (0.63) HPGDSGABRA5CYP2C9MAPK14MAPK11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2307377-A1 NICOTINAMIDE DERIVATIVES Pfizer Limited (GB) 2011-04-13 EP disclosed
WO-2009153720-A1 NICOTINAMIDE DERIVATIVES PFIZER LIMITED (GB) 2009-12-23 WO disclosed