SCHEMBL1543073

SCHEMBL1543073

CC(C(=O)O)[C@H]1CC[C@@H](NC(=O)c2ccc(-c3cccc(F)c3)nc2)CC1

nearest known ligand 0.61

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HPGDS O60760 5/20 0.61
GABRA5 P31644 4/20 0.51
MAP4K4 O95819 2/20 0.48
CYP2C9 P11712 5/20 0.48
MAPK14 Q16539 5/20 0.48
MAPK11 Q15759 1/20 0.47
GRM5 P41594 1/20 0.47
WNT3A P56704 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1543076 1.00 HPGDS (0.61) HPGDSGABRA5MAP4K4CYP2C9MAPK14
SCHEMBL2986337 0.90 HPGDS (0.63) HPGDSGABRA5MAP4K4CYP2C9MAPK14
SCHEMBL13240674 0.90 HPGDS (0.63) HPGDSGABRA5MAP4K4CYP2C9MAPK14
SCHEMBL2986340 0.90 HPGDS (0.63) HPGDSGABRA5MAP4K4CYP2C9MAPK14
SCHEMBL1543340 0.89 HPGDS (0.74) HPGDSGABRA5MAP4K4CYP2C9MAPK14
SCHEMBL1543021 0.88 HPGDS (0.65) HPGDSGABRA5MAP4K4CYP2C9MAPK14
SCHEMBL1543334 0.88 HPGDS (0.65) HPGDSGABRA5MAP4K4CYP2C9MAPK14
SCHEMBL1543023 0.88 HPGDS (0.65) HPGDSGABRA5MAP4K4CYP2C9MAPK14
SCHEMBL1543337 0.88 HPGDS (0.65) HPGDSGABRA5MAP4K4CYP2C9MAPK14
SCHEMBL13240700 0.88 HPGDS (0.65) HPGDSGABRA5MAP4K4CYP2C9MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2307377-A1 NICOTINAMIDE DERIVATIVES Pfizer Limited (GB) 2011-04-13 EP disclosed