SCHEMBL15435528

SCHEMBL15435528

N#Cc1[nH]cc(C(=O)O)c1-c1ccc([N+](=O)[O-])c(F)c1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SIRT5 Q9NXA8 1/20 0.41
ATM Q13315 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
CASP6 P55212 2/20 0.37
DNA2 P51530 1/20 0.37
CTDSP1 Q9GZU7 1/20 0.37
DTYMK P23919 1/20 0.36
EIF4E P06730 5/20 0.36
PRKAB2 O43741 5/20 0.36
PRKAG1 P54619 5/20 0.36
PRKAA2 P54646 5/20 0.36
PRKAA1 Q13131 5/20 0.36
PRKAG3 Q9UGI9 5/20 0.36
PRKAG2 Q9UGJ0 5/20 0.36
PRKAB1 Q9Y478 5/20 0.36
CTSK P43235 1/20 0.35
FBP1 P09467 1/20 0.35
SRD5A2 P31213 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL276542 0.85 ALDH1A1 (0.39) ATM
SCHEMBL762317 0.84 ATM (0.33) SIRT5ATMTDP1CTSK
SCHEMBL10123687 0.78 PDGFRB (0.39) ATMTDP1CTSKSRD5A2
SCHEMBL12909115 0.75 ATM (0.35) ATMTDP1
SCHEMBL27663200 0.72 ATM (0.32) ATMTDP1
SCHEMBL744523 0.72 POLB (0.42)
SCHEMBL762777 0.71 TSHR (0.33)
SCHEMBL10225351 0.70 TDP1 (0.38) SIRT5ATMTDP1FBP1
SCHEMBL3614741 0.68 AR (0.40) ATM
SCHEMBL275419 0.68 MAPT (0.41) ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1957077-B1 SUBSTITUTED 4-AMINO-PYRROLOTRIAZINE DERIVATIVES USEFUL FOR TREATING HYPER-PROLIFERATIVE DISORDERS AND DISEASES ASSOCIATED WITH ANGIOGENESIS BAYER HEALTHCARE LLC (US) 2014-01-22 EP disclosed