SCHEMBL15436288

SCHEMBL15436288

CCC(C(=O)O)c1c2n(c3c(F)cccc13)C[C@H](N=[N+]=[N-])CC2

nearest known ligand 0.39

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PTGDR Q13258 5/20 0.39
PTGDR2 Q9Y5Y4 5/20 0.39
TBXA2R P21731 4/20 0.39
CYP2C9 P11712 2/20 0.39
DPP7 Q9UHL4 2/20 0.33
DPP8 Q6V1X1 1/20 0.33
DPP9 Q86TI2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15006653 0.84 PTGDR2 (0.44) PTGDRPTGDR2TBXA2RCYP2C9
SCHEMBL15436290 0.82 TBXA2R (0.38) PTGDRPTGDR2TBXA2RCYP2C9
SCHEMBL2187304 0.75 PTGDR2 (0.40) PTGDRPTGDR2TBXA2RCYP2C9
SCHEMBL15436289 0.72
SCHEMBL12002786 0.70 CYP2C9 (0.36) PTGDRPTGDR2TBXA2RCYP2C9
SCHEMBL12002746 0.68 PTGDR (0.36) PTGDRPTGDR2TBXA2RCYP2C9
SCHEMBL15436295 0.66 PTGDR2 (0.55) PTGDRPTGDR2TBXA2RCYP2C9
SCHEMBL15436636 0.66 PTGDR2 (0.55) PTGDRPTGDR2TBXA2RCYP2C9
SCHEMBL15436284 0.65 CYP2C9 (0.33) PTGDRPTGDR2TBXA2RCYP2C9
SCHEMBL15165873 0.65 AKR1C3 (0.45)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2401269-B1 INDOLE DERIVATIVES AS CRTH2 RECEPTOR ANTAGONISTS MERCK SHARP & DOHME (US) 2014-01-29 EP disclosed