SCHEMBL15445016

SCHEMBL15445016

CC1=C(Cc2ccc(F)cc2)NNN1C1CCc2c(CC(=O)O)c3cccc(F)c3n2C1

nearest known ligand 0.55

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 20/20 0.55
PTGDR Q13258 9/20 0.55
TBXA2R P21731 7/20 0.55
CYP2C9 P11712 4/20 0.55
CYP3A4 P08684 2/20 0.41
DRD2 P14416 1/20 0.41
GABRA1 P14867 1/20 0.41
ADRA1D P25100 1/20 0.41
SLC6A3 Q01959 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3090467 0.80 PTGDR2 (0.54) PTGDR2PTGDRTBXA2RCYP2C9CYP3A4
SCHEMBL3083458 0.80 PTGDR2 (0.54) PTGDR2PTGDRTBXA2RCYP2C9CYP3A4
SCHEMBL204983 0.78 PTGDR2 (0.53) PTGDR2PTGDRTBXA2RCYP2C9CYP3A4
SCHEMBL15025403 0.78 PTGDR2 (0.53) PTGDR2PTGDRTBXA2RCYP2C9CYP3A4
SCHEMBL3089889 0.78 PTGDR2 (0.53) PTGDR2PTGDRTBXA2RCYP2C9CYP3A4
SCHEMBL15428828 0.74 PTGDR2 (0.60) PTGDR2PTGDRTBXA2RCYP2C9CYP3A4
SCHEMBL3088522 0.73 PTGDR2 (0.64) PTGDR2PTGDRTBXA2RCYP2C9CYP3A4
SCHEMBL3085507 0.72 PTGDR2 (0.49) PTGDR2PTGDRTBXA2RCYP2C9
SCHEMBL3091558 0.71 PTGDR2 (0.54) PTGDR2PTGDRTBXA2RCYP2C9CYP3A4
SCHEMBL3099692 0.71 PTGDR2 (0.46) PTGDR2PTGDRTBXA2RCYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2401269-B1 INDOLE DERIVATIVES AS CRTH2 RECEPTOR ANTAGONISTS MERCK SHARP & DOHME (US) 2014-01-29 EP disclosed