SCHEMBL15463569

SCHEMBL15463569

CC(NC(=O)c1cc(Cl)cnc1COc1ccc(Cl)cc1)c1ccc(C(=O)O)cc1

nearest known ligand 0.73

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PTGER4 P35408 19/20 0.73
PTGER2 P43116 6/20 0.64
RXRA P19793 1/20 0.47
RXRB P28702 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL691834 1.00 PTGER4 (0.73) PTGER4PTGER2RXRARXRB
SCHEMBL3983551 0.93 PTGER4 (0.75) PTGER4PTGER2
SCHEMBL15463534 0.93 PTGER4 (0.75) PTGER4PTGER2
SCHEMBL22076506 0.91 PTGER4 (0.64) PTGER4PTGER2
SCHEMBL692562 0.91 PTGER4 (0.64) PTGER4PTGER2
SCHEMBL3978649 0.91 PTGER4 (0.61) PTGER4PTGER2
SCHEMBL690945 0.89 PTGER4 (0.75) PTGER4PTGER2RXRARXRB
SCHEMBL5502232 0.89 PTGER4 (0.75) PTGER4PTGER2RXRARXRB
SCHEMBL27681503 0.87 PTGER4 (0.56) PTGER4PTGER2RXRARXRB
SCHEMBL3981739 0.87 PTGER4 (0.76) PTGER4PTGER2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102421429-A Selective EP4 receptor antagonist for cancer therapy RAQUALIA PHARMA INC 2012-04-18 CN claimed
CN-1950333-A Substituted methyl aryl or heteroaryl amide compounds PFIZER (US) 2007-04-18 CN claimed
EP-1756042-B1 SUBSTITUTED METHYL ARYL OR HETEROARYL AMIDE COMPOUNDS RAQUALIA PHARMA INC (JP) 2014-02-12 EP disclosed
CN-102770159-A Use of EP-4 receptor antagonists for the treatment of IL-23 mediated diseases RAQUALIA PHARMA INC 2012-11-07 CN disclosed
CN-102421429-A Selective EP4 receptor antagonist for cancer therapy RAQUALIA PHARMA INC 2012-04-18 CN disclosed
CN-1950333-A Substituted methyl aryl or heteroaryl amide compounds PFIZER (US) 2007-04-18 CN disclosed
CN-1946391-A Combinations comprising alpha-2-delta ligands PFIZER PROD INC (US) 2007-04-11 CN disclosed