SCHEMBL15468574

SCHEMBL15468574

CC(C)(C)COC(=O)N(C(=O)OC(C)(C)C)c1ncccc1-c1cc(Cc2ccc(COc3ccccn3)cc2)no1

nearest known ligand 0.33

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 1/20 0.33
HPGD P15428 2/20 0.32
MAPT P10636 1/20 0.32
NPY1R P25929 1/20 0.32
NPY2R P49146 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
BRD4 O60885 1/20 0.32
MCHR1 Q99705 1/20 0.31
ALDH1A1 P00352 3/20 0.31
CYP2C19 P33261 3/20 0.31
CYP1A2 P05177 2/20 0.31
POLB P06746 1/20 0.31
CYP2C9 P11712 1/20 0.31
NPC1 O15118 2/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2D6 P10635 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1322724 0.94 PPARA (0.35) PPARAHPGDMAPTNPY1RNPY2R
SCHEMBL30025507 0.84 CYP11B1 (0.33) PPARAMAPT
SCHEMBL2949533 0.83 ALDH1A1 (0.39) PPARAHPGDMAPTNPY1RNPY2R
SCHEMBL13017182 0.82 MAOB (0.41) PPARAHPGDMAPTSMN1; SMN2BRD4
SCHEMBL26297255 0.82 MAPT (0.37) PPARAHPGDMAPTSMN1; SMN2ALDH1A1
SCHEMBL2303739 0.80 ALDH1A1 (0.37) PPARASMN1; SMN2BRD4MCHR1ALDH1A1
SCHEMBL30025345 0.80 PPARA (0.35) PPARAHPGDSMN1; SMN2ALDH1A1CYP1A2
SCHEMBL13784389 0.78 HPGD (0.36) PPARAHPGDMAPTNPY1RNPY2R
SCHEMBL3422458 0.78 ALDH1A1 (0.37) PPARAHPGDMAPTNPY1RNPY2R
SCHEMBL30025944 0.77 BRS3 (0.34) PPARAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2223926-B1 PYRIDINE DERIVATIVE SUBSTITUTED WITH HETEROCYCLE AND PHOSPHONOXYMETHYL GROUP AND ANTIFUNGAL AGENT CONTAINING THE SAME EISAI R&D MAN CO LTD (JP) 2014-02-12 EP disclosed