SCHEMBL15501243

SCHEMBL15501243

NNC(=O)c1cc(Oc2ccc(NC(=O)CC(=O)Nc3cccc(OC(F)(F)F)c3)cc2)ccn1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAF1 P04049 7/20 0.59
EPHX2 P34913 2/20 0.59
BRAF P15056 7/20 0.57
KDR P35968 5/20 0.57
RET P07949 3/20 0.55
PLK4 O00444 2/20 0.55
AURKA O14965 2/20 0.55
MAPK13 O15264 2/20 0.55
MAP4K4 O95819 2/20 0.55
ABL1 P00519 2/20 0.55
LCK P06239 2/20 0.55
FYN P06241 2/20 0.55
LYN P07948 2/20 0.55
SRC P12931 2/20 0.55
RPS6KB1 P23443 2/20 0.55
EPHA2 P29317 2/20 0.55
AXL P30530 2/20 0.55
FRK P42685 2/20 0.55
MAPK9 P45984 2/20 0.55
BLK P51451 2/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14422934 0.91 RAF1 (0.72) RAF1EPHX2BRAFKDRRET
SCHEMBL14422927 0.87 RAF1 (0.65) RAF1EPHX2BRAFKDRRET
SCHEMBL14422926 0.80 KDR (0.71) RAF1EPHX2BRAFKDRRET
SCHEMBL14422929 0.79 KDR (0.85) RAF1EPHX2BRAFKDRRET
SCHEMBL14422924 0.77 KDR (0.75) RAF1EPHX2BRAFKDRRET
SCHEMBL14022017 0.76 BRAF (0.72) RAF1EPHX2BRAFKDRMAPK14
SCHEMBL14422932 0.75 KDR (0.70) RAF1EPHX2BRAFKDRRET
SCHEMBL5635415 0.75 RET (0.86) RAF1EPHX2BRAFKDRRET
SCHEMBL15624828 0.74 RAF1 (1.00) RAF1EPHX2BRAFKDRRET
SCHEMBL2748558 0.74 KDR (0.56) BRAFKDRRETPDGFRBKIT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1641759-B1 MALONAMIDE DERIVATIVES MERCK PATENT GMBH (DE) 2014-03-12 EP disclosed