SCHEMBL15512970

SCHEMBL15512970

CC(=O)CCCCC[C@H](NC(=O)Cc1c[nH]c2cc(F)ccc12)c1ncc(-c2ccccc2)[nH]1

nearest known ligand 0.60

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 18/20 0.60
HDAC3 O15379 4/20 0.60
HDAC2 Q92769 2/20 0.60
HDAC4 P56524 1/20 0.60
HDAC6 Q9UBN7 1/20 0.60
SSTR1 P30872 2/20 0.52
SSTR3 P32745 2/20 0.52
SSTR5 P35346 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL2074374 0.96 HDAC1 (0.56) HDAC1HDAC3HDAC2HDAC4HDAC6
SCHEMBL15513297 0.94 HDAC1 (0.62) HDAC1HDAC3HDAC2HDAC4HDAC6
Trifluoroacetic Acid SCHEMBL2070991 0.90 HDAC1 (0.58) HDAC1HDAC3HDAC2HDAC4HDAC6
SCHEMBL15513687 0.90 HDAC1 (0.63) HDAC1HDAC3HDAC2HDAC4HDAC6
Trifluoroacetic Acid SCHEMBL2071490 0.88 HDAC1 (0.58) HDAC1HDAC3HDAC2HDAC4HDAC6
SCHEMBL15512872 0.87 HDAC1 (0.62) HDAC1HDAC3HDAC2HDAC4HDAC6
SCHEMBL15513177 0.86 HDAC1 (0.62) HDAC1HDAC3HDAC2HDAC4HDAC6
SCHEMBL15514020 0.86 HDAC1 (0.62) HDAC1HDAC3HDAC2HDAC4HDAC6
SCHEMBL15512867 0.85 HDAC1 (0.76) HDAC1HDAC3HDAC2HDAC4HDAC6
Trifluoroacetic Acid SCHEMBL2070841 0.84 HDAC1 (0.58) HDAC1HDAC3HDAC2HDAC4HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1828171-B1 HETEROCYCLE DERIVATIVES AS HISTONE DEACETYLASE (HDAC) INHIBITORS ANGELETTI P IST RICHERCHE BIO (IT) 2014-03-12 EP claimed