SCHEMBL15515696

SCHEMBL15515696

NC(=O)c1cccc(-c2cc3c(N4CCN(c5ccc(OC(F)(F)F)cc5)CC4)ncnc3[nH]2)c1

nearest known ligand 0.79

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
KIT P10721 20/20 0.79

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15515316 0.91 KIT (0.80) KIT
SCHEMBL15663671 0.88 KIT (1.00) KIT
SCHEMBL15515575 0.85 KIT (0.82) KIT
SCHEMBL15515978 0.83 KIT (0.62) KIT
SCHEMBL15515827 0.83 KIT (0.79) KIT
SCHEMBL15664565 0.80 KIT (1.00) KIT
SCHEMBL15664520 0.79 KIT (1.00) KIT
SCHEMBL15516953 0.79 KIT (0.75) KIT
SCHEMBL15515412 0.77 KIT (0.79) KIT
SCHEMBL15516553 0.77 KIT (0.75) KIT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2892534-A2 COMPOUNDS AND METHODS FOR KINASE MODULATION, AND INDICATIONS THEREFOR Plexxikon, Inc. (US) 2015-07-15 EP disclosed
WO-2014039714-A2 COMPOUNDS AND METHODS FOR KINASE MODULATION, AND INDICATIONS THEREFOR PLEXXIKON INC. (US) 2014-03-13 WO disclosed