SCHEMBL1551653

SCHEMBL1551653

NC(=O)Oc1ccc2[nH]c(-c3ccc(OCCC4CCNCC4)cc3)nc2c1

nearest known ligand 0.70

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 17/20 0.70
DHODH Q02127 1/20 0.58
ADORA3 P0DMS8 1/20 0.50
ADORA2A P29274 1/20 0.50
ADORA2B P29275 1/20 0.50
ADORA1 P30542 1/20 0.50
ITGB3 P05106 1/20 0.47
ITGA2B P08514 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1552741 0.90 CHEK2 (0.69) CHEK2DHODH
SCHEMBL1551751 0.88 CHEK2 (0.85) CHEK2DHODH
SCHEMBL1551713 0.87 CHEK2 (0.73) CHEK2DHODH
SCHEMBL5176542 0.86 CHEK2 (0.53) CHEK2DHODH
SCHEMBL1552651 0.85 CHEK2 (0.72) CHEK2
SCHEMBL1552385 0.85 CHEK2 (0.77) CHEK2DHODH
SCHEMBL1553042 0.85 CHEK2 (0.67) CHEK2
SCHEMBL1552781 0.84 CHEK2 (0.65) CHEK2DHODH
SCHEMBL1552763 0.84 CHEK2 (0.74) CHEK2
SCHEMBL1551654 0.84 CHEK2 (0.75) CHEK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1824832-B1 ARYL-SUBSTITUTED BENZIMIDAZOLE AND IMIDAZOPYRIDINE ETHERS AS ANTI-CANCER AGENTS JANSSEN PHARMACEUTICA NV (BE) 2011-04-27 EP claimed