SCHEMBL15519642

SCHEMBL15519642

CC(c1ccc(-c2ccc(OC(=O)O)cc2)cc1Cl)C(O)(c1ccc2c(c1)N(C)C(=O)CO2)C(F)(F)F

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GPR55 Q9Y2T6 1/20 0.37
ALDH1A1 P00352 1/20 0.35
PDE3B Q13370 1/20 0.34
PDE3A Q14432 1/20 0.34
CTSC P53634 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
BRD4 O60885 1/20 0.32
KMO O15229 2/20 0.32
USP2 O75604 1/20 0.32
HTT P42858 1/20 0.32
CYP11B1 P15538 1/20 0.31
CYP11B2 P19099 1/20 0.31
POLB P06746 1/20 0.31
ESR1 P03372 1/20 0.31
CYP3A4 P08684 4/20 0.31
CYP2D6 P10635 4/20 0.31
OPRK1 P41145 4/20 0.31
UTS2R Q9UKP6 4/20 0.31
THRB P10828 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15520696 0.94 GPR55 (0.37) GPR55ALDH1A1PDE3BPDE3ACTSC
SCHEMBL15520294 0.93 GPR55 (0.36) GPR55ALDH1A1PDE3BPDE3AKMO
SCHEMBL15520371 0.92 GPR55 (0.37) GPR55ALDH1A1PDE3BPDE3ACTSC
SCHEMBL15520206 0.91 GPR55 (0.37) GPR55ALDH1A1PDE3BPDE3ACTSC
SCHEMBL15520365 0.91 FFAR4 (0.35) GPR55ALDH1A1PDE3BPDE3AKMO
SCHEMBL15520588 0.91 GPR55 (0.35) GPR55ALDH1A1PDE3BPDE3AESR1
SCHEMBL15520752 0.91 GPR55 (0.38) GPR55ALDH1A1PDE3BPDE3ACTSC
SCHEMBL15520803 0.91 GPR55 (0.38) GPR55ALDH1A1PDE3BPDE3ACTSC
SCHEMBL15520533 0.91 GPR55 (0.38) GPR55ALDH1A1PDE3BPDE3ACTSC
SCHEMBL473952 0.90 GPR55 (0.39) GPR55ALDH1A1PDE3BPDE3ACTSC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411365-B1 2,3-DIARYL- OR HETEROARYL-SUBSTITUTED 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS HOFFMANN LA ROCHE (CH) 2014-03-19 EP claimed