SCHEMBL15519977

SCHEMBL15519977

CCN(C[C@H]1CC[C@H](CC(=O)O)CC1)c1ncc(C(F)(F)F)cc1CN(CCc1cc(C(F)(F)F)cc(C(F)(F)F)c1)[SH](=O)=O

nearest known ligand 0.34

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 8/20 0.34
CYP3A4 P08684 6/20 0.34
DGAT1 O75907 4/20 0.33
FFAR4 Q5NUL3 3/20 0.33
KCNH2 Q12809 2/20 0.33
ADORA2A P29274 1/20 0.33
PTGDR2 Q9Y5Y4 1/20 0.33
TRPM8 Q7Z2W7 1/20 0.33
LTC4S Q16873 1/20 0.32
HTR1A P08908 1/20 0.32
ADRA2A P08913 1/20 0.32
ADRA1A P35348 1/20 0.32
HTR2B P41595 1/20 0.32
MCHR1 Q99705 1/20 0.32
SOAT1 P35610 1/20 0.32
RORC P51449 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL680558 0.85 GPBAR1 (0.44) TACR1CYP3A4DGAT1FFAR4KCNH2
SCHEMBL680559 0.85 GPBAR1 (0.44) TACR1CYP3A4DGAT1FFAR4KCNH2
SCHEMBL680455 0.83 TACR1 (0.39) TACR1CYP3A4DGAT1KCNH2ADORA2A
SCHEMBL680456 0.83 TACR1 (0.39) TACR1CYP3A4DGAT1KCNH2ADORA2A
SCHEMBL680976 0.83 TACR1 (0.36) TACR1CYP3A4DGAT1FFAR4KCNH2
SCHEMBL679436 0.83 GPBAR1 (0.36) TACR1CYP3A4DGAT1FFAR4KCNH2
SCHEMBL679435 0.83 GPBAR1 (0.36) TACR1CYP3A4DGAT1FFAR4KCNH2
SCHEMBL680262 0.83 CETP (0.46) PTGDR2
SCHEMBL680263 0.83 CETP (0.46) PTGDR2
SCHEMBL680975 0.81 TRPM8 (0.34) TACR1CYP3A4DGAT1FFAR4KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2383253-B1 METHOD FOR MANUFACTURING TRANS-{4-[(ALKYL AMINO) METHYL]CYCLOHEXYL} ACETIC ESTER KOWA CO (JP) 2014-03-19 EP disclosed