SCHEMBL15529385

SCHEMBL15529385

NC1C(C(=O)O)[C@H]2C=C[C@@H]1C2

nearest known ligand 0.65

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.65
CYP2C19 P33261 1/20 0.65
POLB P06746 5/20 0.50
TDP1 Q9NUW8 3/20 0.50
APEX1 P27695 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.43
GAA P10253 1/20 0.41
NPSR1 Q6W5P4 1/20 0.39
TAAR1 Q96RJ0 1/20 0.39
CASP6 P55212 1/20 0.39
CTDSP1 Q9GZU7 1/20 0.39
HSD17B10 Q99714 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1484126 1.00 ALDH1A1 (0.65) ALDH1A1CYP2C19POLBTDP1APEX1
SCHEMBL2033299 1.00 ALDH1A1 (0.65) ALDH1A1CYP2C19POLBTDP1APEX1
SCHEMBL7232865 1.00 ALDH1A1 (0.65) ALDH1A1CYP2C19POLBTDP1APEX1
SCHEMBL311527 1.00 ALDH1A1 (0.65) ALDH1A1CYP2C19POLBTDP1APEX1
Hydrochloric Acid SCHEMBL26613189 0.98 ALDH1A1 (0.63) ALDH1A1CYP2C19POLBTDP1APEX1
Hydrochloric Acid SCHEMBL26613207 0.98 ALDH1A1 (0.63) ALDH1A1CYP2C19POLBTDP1APEX1
Hydrochloric Acid SCHEMBL19668549 0.98 ALDH1A1 (0.63) ALDH1A1CYP2C19POLBTDP1APEX1
Hydrochloric Acid SCHEMBL19668550 0.98 ALDH1A1 (0.63) ALDH1A1CYP2C19POLBTDP1APEX1
SCHEMBL24062391 0.83 POLB (0.70) ALDH1A1POLBTDP1APEX1SMN1; SMN2
SCHEMBL20346210 0.83 POLB (0.70) ALDH1A1POLBTDP1APEX1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 43 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024130161-A2 NOVEL CAMPTOTHECIN DERIVATIVES AND CONJUGATES THEREOF BIONECURE THERAPEUTICS INC (US) 2024-06-20 WO disclosed
US-20240034753-A1 THERAPEUTIC PEPTIDES COHBAR, INC. 2024-02-01 US disclosed
US-11753445-B2 Therapeutic peptides COHBAR, INC. (US) 2023-09-12 US disclosed
US-20230218710-A1 METHOD OF TREATING CORONAVIRUS INFECTIONS COHBAR, INC. 2023-07-13 US disclosed
US-20230137562-A1 TAU AGGREGATION INHIBITORS ADRX, INC. 2023-05-04 US disclosed
EP-4135738-A2 METHOD OF TREATING CORONAVIRUS INFECTIONS Cohbar Inc. (US) 2023-02-22 EP disclosed
US-20220395553-A1 CXCR4 ANTAGONIST PEPTIDES COHBAR, INC. 2022-12-15 US disclosed
US-20220332774-A1 THERAPEUTIC MITOCHONDRIAL PEPTIDES COHBAR, INC. 2022-10-20 US disclosed
US-20220324909-A1 THERAPEUTIC PEPTIDES COHBAR, INC. 2022-10-13 US disclosed
US-20220324925-A1 THERAPEUTIC PEPTIDES COHBAR, INC. 2022-10-13 US disclosed
US-20200216495-A1 TAU AGGREGATION PEPTIDE INHIBITORS ADRX, INC. 2020-07-09 US disclosed
EP-3668886-A2 TAU AGGREGATION PEPTIDE INHIBITORS Adrx, Inc. (US) 2020-06-24 EP disclosed
US-20200181197-A1 THERAPEUTIC PEPTIDES COHBAR, INC. 2020-06-11 US disclosed
US-20200062804-A1 PEPTIDE INHIBITORS OF TRANSCRIPTION FACTOR AGGREGATION ADRX, INC. 2020-02-27 US disclosed
EP-3519431-A1 THERAPEUTIC MOTS-C RELATED PEPTIDES Cohbar Inc. (US) 2019-08-07 EP disclosed
WO-2019036725-A2 TAU AGGREGATION PEPTIDE INHIBITORS ADRX, INC. (US) 2019-02-21 WO disclosed
WO-2018156892-A1 PEPTIDE INHIBITORS OF TRANSCRIPTION FACTOR AGGREGATION ADRX, INC. (US) 2018-08-30 WO disclosed
WO-2018064098-A1 THERAPEUTIC MOTS-C RELATED PEPTIDES COHBAR, INC. (US) 2018-04-05 WO disclosed
US-20150218538-A1 Methods and Compositions for Modulating G-Alpha-Q Signaling NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2015-08-06 US disclosed
WO-2013165554-A1 METHODS AND COMPOSITIONS FOR MODULATING G-ALPHA-Q SIGNALING THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 2013-11-07 WO disclosed