SCHEMBL15529643

SCHEMBL15529643

O=C(Nc1cccnc1)N1CCC1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 1/20 0.60
FAAH O00519 4/20 0.57
HTR2C P28335 3/20 0.57
GRIN2B Q13224 2/20 0.56
NPC1 O15118 1/20 0.54
PKM P14618 1/20 0.54
RAB9A P51151 1/20 0.54
LMNA P02545 1/20 0.53
HIF1A Q16665 1/20 0.53
HTR2A P28223 2/20 0.52
HDAC3 O15379 1/20 0.52
HDAC1 Q13547 1/20 0.52
HDAC2 Q92769 1/20 0.52
PDGFRB P09619 1/20 0.52
NAMPT P43490 1/20 0.51
ALDH1A1 P00352 2/20 0.51
MEN1 O00255 1/20 0.51
RECQL P46063 1/20 0.51
KMT2A Q03164 1/20 0.51
NPSR1 Q6W5P4 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1960679 0.95 TRPV1 (0.58) TRPV1FAAHHTR2CGRIN2BNPC1
Hydrochloric Acid SCHEMBL2197351 0.94 TRPV1 (0.57) TRPV1FAAHHTR2CGRIN2BNPC1
SCHEMBL3768246 0.88 TRPV1 (0.60) TRPV1FAAHHTR2CGRIN2BNPC1
SCHEMBL30791537 0.86 POLB (0.66) TRPV1FAAHHTR2CGRIN2BNPC1
SCHEMBL1758868 0.86 POLB (0.66) TRPV1FAAHHTR2CGRIN2BNPC1
SCHEMBL6304805 0.85 HTR2C (0.70) TRPV1FAAHHTR2CGRIN2BNPC1
Hydrochloric Acid SCHEMBL2194067 0.85 POLB (0.68) TRPV1FAAHHTR2CGRIN2BNPC1
SCHEMBL32668648 0.85 GRIN2B (0.55) TRPV1FAAHHTR2CGRIN2BLMNA
SCHEMBL16707623 0.84 LMNA (0.67) TRPV1FAAHHTR2CLMNAHTR2A
SCHEMBL12509405 0.83 CYP3A4 (0.63) TRPV1FAAHGRIN2BNPC1PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2852585-A1 NAMPT INHIBITORS AbbVie Inc. (US) 2015-04-01 EP disclosed
WO-2013170113-A1 NAMPT INHIBITORS ABBVIE INC. (US) 2013-11-14 WO disclosed