SCHEMBL15533294

SCHEMBL15533294

COc1ccc(-c2cc(Cl)ncn2)c(OC)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 6/20 0.50
CYP3A4 P08684 6/20 0.50
CYP2D6 P10635 6/20 0.50
CYP2C19 P33261 5/20 0.50
TSHR P16473 5/20 0.50
MAPK1 P28482 4/20 0.50
CLK4 Q9HAZ1 4/20 0.50
MEN1 O00255 4/20 0.50
KMT2A Q03164 4/20 0.50
CYP1A1 P04798 3/20 0.50
CYP1B1 Q16678 3/20 0.50
HSD17B10 Q99714 2/20 0.50
USP2 O75604 1/20 0.50
ALOX15 P16050 1/20 0.50
CYP2E1 P05181 1/20 0.46
CYP2C8 P10632 1/20 0.46
CYP2A6 P11509 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP4B1 P13584 1/20 0.46
CYP2B6 P20813 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30777916 0.83 CYP1A2 (0.48) CYP1A2CYP3A4CYP2D6CYP2C19TSHR
SCHEMBL513403 0.83 KIT (0.45) CYP1A2CYP3A4CYP2D6CYP2C19TSHR
SCHEMBL8514899 0.83 CYP1A2 (0.48) CYP1A2CYP3A4CYP2D6CYP2C19TSHR
SCHEMBL1850151 0.81 HSP90AA1 (0.59) CYP1A2CYP3A4CYP2D6CYP2C19TSHR
SCHEMBL20210912 0.80 SCN9A (0.48) CYP2D6CYP2C19TSHRMAPK1USP2
SCHEMBL511711 0.77 HTT (0.49) CYP1A2CYP3A4CYP2D6CYP2C19MAPK1
SCHEMBL4438489 0.77 CYP1A1 (0.52) MAPK1KMT2ACYP1A1CYP1B1LMNA
SCHEMBL15486382 0.74 CDK9 (0.49) CYP1A2CYP3A4CYP2D6CYP2C19TSHR
SCHEMBL2993281 0.74 HSP90AA1 (0.44) CYP1A2CYP3A4CYP2D6CYP2C19TSHR
SCHEMBL444455 0.74 CYP1A1 (0.52) CYP1A2CYP3A4CYP2D6CYP2C19TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013175415-A1 SUBSTITUTED PYRIMIDINE COMPOUNDS AND USES THEREOF Piramal Enterprises Limited (IN) 2013-11-28 WO disclosed