SCHEMBL15543403

SCHEMBL15543403

[2H]C([2H])(c1ccc(-c2ccc3cc[nH]c3c2)cc1)N1CCC2(CC1)CN(C1CC1)C(=O)CO2

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
FASN P49327 6/20 0.47
KDM4E B2RXH2 2/20 0.34
ALDH1A1 P00352 2/20 0.34
HSD17B10 Q99714 2/20 0.34
SIGMAR1 Q99720 5/20 0.34
OPRM1 P35372 3/20 0.34
CTSC P53634 1/20 0.33
KCNH2 Q12809 1/20 0.33
BACE1 P56817 2/20 0.32
MAPT P10636 1/20 0.30
HPGD P15428 1/20 0.30
MCHR1 Q99705 1/20 0.30
EPHX1 P07099 1/20 0.30
CYP2D6 P10635 1/20 0.30
EPHX2 P34913 1/20 0.30
CREBBP Q92793 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15581799 0.91 FASN (0.48) FASNKDM4EALDH1A1HSD17B10SIGMAR1
SCHEMBL15556185 0.88 FASN (0.43) FASNKDM4EALDH1A1HSD17B10SIGMAR1
Trifluoroacetic Acid SCHEMBL15544054 0.84 FASN (0.43) FASNKDM4EALDH1A1HSD17B10SIGMAR1
Trifluoroacetic Acid SCHEMBL15556665 0.83 FASN (0.39) FASNKDM4EALDH1A1HSD17B10CTSC
SCHEMBL15555919 0.82 FASN (0.46) FASNKDM4EALDH1A1HSD17B10SIGMAR1
SCHEMBL15544258 0.82 FASN (0.44) FASNKDM4EALDH1A1HSD17B10SIGMAR1
SCHEMBL15556670 0.82 FASN (0.44) FASNKDM4EALDH1A1HSD17B10SIGMAR1
SCHEMBL15555329 0.82 FASN (0.44) FASNKDM4EALDH1A1HSD17B10SIGMAR1
SCHEMBL15543680 0.82 FASN (0.70) FASNSIGMAR1OPRM1KCNH2
SCHEMBL4560675 0.81 FASN (0.70) FASNALDH1A1HSD17B10HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014008223-A2 FATTY ACID SYNTHASE INHIBITORS GLAXOSMITHKLINE LLC (US) 2014-01-09 WO claimed
WO-2014008223-A2 FATTY ACID SYNTHASE INHIBITORS GLAXOSMITHKLINE LLC (US) 2014-01-09 WO disclosed