SCHEMBL15544299

SCHEMBL15544299

O=C1CC(c2cc(O)c(O)c(O)c2)Oc2cc(O)cc(O)c21

nearest known ligand 0.83

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TTR P02766 4/20 0.78
CYP19A1 P11511 7/20 0.75
CYP3A4 P08684 6/20 0.75
CYP1A1 P04798 6/20 0.75
CYP1A2 P05177 6/20 0.75
CYP1B1 Q16678 6/20 0.75
CYP2C19 P33261 4/20 0.75
HSD17B10 Q99714 4/20 0.75
CA12 O43570 3/20 0.75
CA4 P22748 3/20 0.75
CA7 P43166 3/20 0.75
MAPT P10636 3/20 0.75
TP53 P04637 3/20 0.75
SLCO2B1 O94956 2/20 0.75
PSMB5 P28074 2/20 0.75
ALDH1A1 P00352 2/20 0.75
PKM P14618 2/20 0.75
HPGD P15428 2/20 0.75
MAPK1 P28482 2/20 0.75
POLB P06746 2/20 0.75

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29991657 1.00 TTR (0.78) TTRCYP19A1CYP3A4CYP1A1CYP1A2
SCHEMBL14374975 1.00 TTR (0.78) TTRCYP19A1CYP3A4CYP1A1CYP1A2
SCHEMBL28616923 0.91 TTR (0.81) TTRCYP19A1CYP3A4CYP1A1CYP1A2
SCHEMBL30689832 0.91 TTR (0.81) TTRCYP19A1CYP3A4CYP1A1CYP1A2
SCHEMBL26130529 0.90 TTR (0.72) TTRCYP19A1CYP3A4CYP1A1CYP1A2
SCHEMBL26406001 0.87 TTR (0.72) TTRCYP19A1CYP3A4CYP1A1CYP1A2
SCHEMBL26128340 0.87 TTR (1.00) TTRCYP19A1CYP3A4CYP1A1CYP1A2
Eriodictyol SCHEMBL23686074 0.86 CYP19A1 (1.00) TTRCYP19A1CYP3A4CYP1A1CYP1A2
Eriodictyol SCHEMBL2309591 0.86 CYP19A1 (1.00) TTRCYP19A1CYP3A4CYP1A1CYP1A2
Eriodictyol SCHEMBL19180 0.86 CYP19A1 (1.00) TTRCYP19A1CYP3A4CYP1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240263203-A1 RECOMBINANT HOST CELLS WITH IMPROVED PRODUCTION OF TETRAKETIDE DERIVATIVES IPTECTOR ASSETS APS (DK) 2024-08-08 US disclosed
WO-2024040211-A2 FLAVONOID BIOPRODUCTION USING MICROORGANISM HOSTS Debut Biotechnology, Inc. (US) 2024-02-22 WO disclosed
EP-4323528-A1 FLAVONOID AND ANTHOCYANIN BIOPRODUCTION USING MICROORGANISM HOSTS Debut Biotechnology, Inc. (US) 2024-02-21 EP disclosed
WO-2022221392-A1 FLAVONOID AND ANTHOCYANIN BIOPRODUCTION USING MICROORGANISM HOSTS Debut Biotechnology, Inc. (US) 2022-10-20 WO disclosed
US-20220257561-A1 COMPOSITIONS AND METHODS FOR IMPROVING WELLNESS ADVANCED DELIVERY LABS LLC (US) 2022-08-18 US disclosed
EP-3906301-A1 RECOMBINANT HOST CELLS WITH IMPROVED PRODUCTION OF TETRAKETIDE DERIVATIVES Barrit Sarl (FR) 2021-11-10 EP disclosed
WO-2020141230-A1 RECOMBINANT HOST CELLS WITH IMPROVED PRODUCTION OF TETRAKETIDE DERIVATIVES BARRIT SARL (FR) 2020-07-09 WO disclosed
US-20190040417-A1 BIOLOGICAL FERMENTATION USING DIHYDROXYACETONE AS A SOURCE OF CARBON KEMBIOTIX LLC (US) 2019-02-07 US disclosed
US-10119154-B2 Anthocyanins with specific properties EVOLVA SA (CH) 2018-11-06 US disclosed
WO-2017139420-A1 BIOLOGICAL FERMENTATION USING DIHYDROXYACETONE AS A SOURCE OF CARBON KEMBIOTIX LLC (US) 2017-08-17 WO disclosed
US-20160319290-A2 NOVEL PROTEIN AND GENE RELATED TO FLAVONOID O-METHYLTRANSFERASE (FOMT) AND THEIR USES THEREFORE INST BOTANY CAS (CN) 2016-11-03 US disclosed
US-20150344920-A1 Anthocyanins with Specific Properties EVOLVA SA (CH) 2015-12-03 US disclosed
EP-2935607-A1 ANTHOCYANINS WITH SPECIFIC PROPERTIES Evolva SA (CH) 2015-10-28 EP disclosed
WO-2014096456-A1 ANTHOCYANINS WITH SPECIFIC PROPERTIES EVOLVA SA (CH) 2014-06-26 WO disclosed
WO-2014007853-A1 DIHYDROMYRICETIN FOR THE TREATMENT OF DISEASES AND DISORDERS OF THE GLUTAMATERGIC SYSTEM THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2014-01-09 WO disclosed