SCHEMBL15553827

SCHEMBL15553827

COc1ccc(-c2cnc3[nH]cc(-c4ccc(OCCN(C)C)c(C#N)c4)c3c2)cc1OC

nearest known ligand 0.66

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KIT P10721 15/20 0.66
DYRK1A Q13627 2/20 0.66
AAK1 Q2M2I8 1/20 0.58
NTRK1 P04629 1/20 0.58
MAP3K11 Q16584 1/20 0.58
PIK3CA P42336 1/20 0.57
SLC2A1 P11166 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15553414 0.90 KIT (0.69) KITDYRK1AAAK1MAP3K11PIK3CA
SCHEMBL15553843 0.88 KIT (0.80) KITDYRK1AAAK1MAP3K11PIK3CA
SCHEMBL722517 0.83 MAP3K11 (0.79) KITDYRK1AAAK1NTRK1MAP3K11
SCHEMBL12763552 0.81 AAK1 (0.62) KITDYRK1AAAK1NTRK1SLC2A1
SCHEMBL15833894 0.81 KIT (1.00) KITDYRK1AAAK1NTRK1PIK3CA
SCHEMBL15560067 0.80 KIT (0.69) KITDYRK1AMAP3K11PIK3CA
SCHEMBL7910200 0.79 KIT (0.58) KITDYRK1AAAK1NTRK1PIK3CA
SCHEMBL15553965 0.79 KIT (0.66) KITDYRK1AAAK1MAP3K11PIK3CA
SCHEMBL15554558 0.78 KIT (0.52) KITNTRK1PIK3CA
SCHEMBL15554959 0.78 MAP4K1 (0.66) KITDYRK1AAAK1MAP3K11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014004863-A2 COMPOUNDS, COMPOSITIONS, AND THERAPEUTIC USES THEREOF ALZHEIMER'S INSTITUTE OF AMERICA, INC. (US) 2014-01-03 WO claimed
WO-2014004863-A2 COMPOUNDS, COMPOSITIONS, AND THERAPEUTIC USES THEREOF ALZHEIMER'S INSTITUTE OF AMERICA, INC. (US) 2014-01-03 WO disclosed