SCHEMBL15566545

SCHEMBL15566545

Cn1nc(C(N)=O)c(N)c1C1CCCC1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 1/20 0.41
CCNA2 P20248 4/20 0.36
CDK2 P24941 4/20 0.36
CCNA1 P78396 4/20 0.36
HPGD P15428 1/20 0.35
RET P07949 1/20 0.33
PDE4D Q08499 2/20 0.32
PDE7A Q13946 2/20 0.32
ALDH1A1 P00352 2/20 0.32
JAK2 O60674 1/20 0.32
JAK1 P23458 1/20 0.32
TYK2 P29597 1/20 0.32
JAK3 P52333 1/20 0.32
MEN1 O00255 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
HTT P42858 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15566566 0.78 SMN1; SMN2 (0.40) GRM5CCNA2CDK2CCNA1HPGD
SCHEMBL3996291 0.71 ALOX5AP (0.33) HPGDRETPDE4DPDE7AALDH1A1
SCHEMBL6385540 0.71 GFER (0.34) CDK8
SCHEMBL7522906 0.70 PIM3 (0.41) CCNA2CDK2CCNA1HPGDALDH1A1
SCHEMBL6386074 0.69 GAA (0.34) CDK8
SCHEMBL7001118 0.68 ADORA2A (0.37) CCNA2CDK2CCNA1HPGDALDH1A1
Bromide SCHEMBL7823529 0.67 ADORA2A (0.36) CCNA2CDK2CCNA1HPGDALDH1A1
SCHEMBL5230043 0.67 RET (0.42) CCNA2CDK2CCNA1RETPDE4D
SCHEMBL1814028 0.67 RET (0.42) CCNA2CDK2CCNA1RETPDE4D
SCHEMBL21501683 0.66 PDE10A (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014024125-A1 PYRAZOLO[4,3-D]PYRIMIDIN-7(6H)-ONE DERIVATIVES AS PDE9 INHIBITORS CELON PHARMA S.A. (PL) 2014-02-13 WO disclosed