SCHEMBL15568136

SCHEMBL15568136

C#CCn1c(-c2ccccc2Br)nc2ccccc21

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.47
TP53 P04637 2/20 0.47
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
MAPT P10636 4/20 0.45
TDP1 Q9NUW8 1/20 0.45
KDM4E B2RXH2 4/20 0.44
LMNA P02545 3/20 0.44
HTT P42858 3/20 0.44
ALDH1A1 P00352 3/20 0.44
TSHR P16473 2/20 0.44
HPGD P15428 1/20 0.44
ALOX15 P16050 1/20 0.44
NPY1R P25929 1/20 0.44
MAPK1 P28482 1/20 0.44
NPY2R P49146 1/20 0.44
HSD17B10 Q99714 1/20 0.44
TLR7 Q9NYK1 1/20 0.42
NPSR1 Q6W5P4 4/20 0.41
GAA P10253 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30581236 0.77 KDM4E (0.60) SMN1; SMN2TP53MEN1KMT2AMAPT
SCHEMBL29076126 0.77 KDM4E (0.60) SMN1; SMN2TP53MEN1KMT2AMAPT
SCHEMBL6810630 0.76 TLR8 (0.57) SMN1; SMN2TP53MEN1KMT2AMAPT
SCHEMBL20421688 0.75 TNF (0.58) SMN1; SMN2TP53MEN1KMT2AMAPT
SCHEMBL21085204 0.74 KDM4E (0.64) SMN1; SMN2TP53MEN1KMT2AMAPT
SCHEMBL1482899 0.73 PRKACA (0.53) TP53KDM4EHTTALDH1A1TSHR
SCHEMBL10061948 0.72 TP53 (0.45) SMN1; SMN2TP53MEN1KMT2AMAPT
SCHEMBL228955 0.72 ALDH1A1 (0.56) SMN1; SMN2TP53MEN1KMT2AMAPT
SCHEMBL10061943 0.71 KDM4E (0.70) SMN1; SMN2TP53MEN1KMT2AMAPT
SCHEMBL23673271 0.71 KDM4E (0.44) SMN1; SMN2TP53MEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014027053-A1 BENZIMIDAZOLES FOR THE TREATMENT OF CANCER MAX-PLANCK-Gesellschaft zur Förderung der Wissenschaften e.V. (DE) 2014-02-20 WO disclosed