SCHEMBL15575223

SCHEMBL15575223

CN(C)CCCOc1ccccc1NC(=O)NCc1ccc(Oc2ccncc2)cc1

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.51
CACNA1B Q00975 8/20 0.51
CACNA1H O95180 3/20 0.51
KMT2A Q03164 2/20 0.51
MEN1 O00255 1/20 0.51
GAA P10253 1/20 0.51
ALDH1A1 P00352 2/20 0.49
NAMPT P43490 1/20 0.47
TRPV1 Q8NER1 1/20 0.46
HDAC1 Q13547 1/20 0.45
HDAC6 Q9UBN7 1/20 0.45
ROCK2 O75116 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2C9 P11712 1/20 0.45
ROCK1 Q13464 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16990731 0.88 CACNA1B (0.48) POLBCACNA1BCACNA1HKMT2AMEN1
SCHEMBL13603469 0.87 DDR2 (0.52) POLBCACNA1BCACNA1HKMT2AMEN1
SCHEMBL15575211 0.83 ALDH1A1 (0.66) POLBKMT2AMEN1GAAALDH1A1
SCHEMBL15575316 0.79 NAMPT (0.61) KMT2AMEN1GAAALDH1A1NAMPT
SCHEMBL15574706 0.78 ALDH1A1 (0.57) POLBKMT2AMEN1GAAALDH1A1
SCHEMBL15574561 0.77 NAMPT (0.61) POLBKMT2AMEN1ALDH1A1NAMPT
SCHEMBL15574732 0.77 ALDH1A1 (0.55) KMT2AMEN1ALDH1A1NAMPTTRPV1
SCHEMBL16990677 0.76 DDR2 (0.74) ALDH1A1NAMPTROCK2CYP3A4CYP2D6
SCHEMBL16990708 0.76 RAF1 (0.58) ALDH1A1TRPV1
SCHEMBL16990698 0.75 NAMPT (0.61) ALDH1A1NAMPTROCK2CYP3A4ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2890380-A2 DDR2 INHIBITORS FOR THE TREATMENT OF OSTEOARTHRITIS Merck Patent GmbH (DE) 2015-07-08 EP disclosed
WO-2014032755-A2 DDR2 INHIBITORS FOR THE TREATMENT OF OSTEOARTHRITIS MERCK PATENT GMBH (DE) 2014-03-06 WO disclosed