SCHEMBL15577609

SCHEMBL15577609

O=CC[C@@H](c1ccc(F)cc1)c1ccccc1F

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.40
HTT P42858 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
ALDH1A1 P00352 2/20 0.38
MEN1 O00255 4/20 0.37
KMT2A Q03164 4/20 0.37
CACNA1B Q00975 2/20 0.37
CACNA2D1 P54289 1/20 0.37
CACNB1 Q02641 1/20 0.37
CACNA1C Q13936 1/20 0.37
IDO1 P14902 1/20 0.37
TDO2 P48775 1/20 0.37
GAA P10253 1/20 0.36
CYP19A1 P11511 2/20 0.36
CNR2 P34972 2/20 0.36
POLB P06746 1/20 0.35
CNR1 P21554 2/20 0.35
CYP2D6 P10635 2/20 0.34
SLC6A2 P23975 2/20 0.34
SLC6A4 P31645 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL65457 0.82 CACNA2D1 (0.37) MAPK1HTTCACNA1BCACNA2D1CACNB1
SCHEMBL15577652 0.78 PTGDR2 (0.39) HTTMEN1KMT2ACYP19A1POLB
Ammonia Solution, Strong SCHEMBL6001428 0.77 HTT (0.40) MAPK1HTTSMN1; SMN2ALDH1A1MEN1
SCHEMBL27506211 0.77 IDO1 (0.40) MAPK1HTTSMN1; SMN2ALDH1A1MEN1
SCHEMBL15577608 0.77 IDO1 (0.40) MAPK1HTTSMN1; SMN2ALDH1A1MEN1
SCHEMBL6001426 0.76 HRH1 (0.53) MAPK1HTTSMN1; SMN2ALDH1A1KMT2A
SCHEMBL15577528 0.75 HTR2A (0.41) MAPK1SMN1; SMN2ALDH1A1MEN1KMT2A
SCHEMBL29791196 0.74 TBXA2R (0.42) ALDH1A1CACNA1BGAACYP19A1CNR2
SCHEMBL30758302 0.74 TBXA2R (0.42) ALDH1A1CACNA1BGAACYP19A1CNR2
SCHEMBL777581 0.74 ALDH1A1 (0.40) ALDH1A1GAACNR2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2895482-A1 HIV PROTEASE INHIBITORS Merck Sharp & Dohme Corp. (US) 2015-07-22 EP disclosed
WO-2014043019-A1 HIV PROTEASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2014-03-20 WO disclosed