SCHEMBL15580688

SCHEMBL15580688

Cc1cc(Oc2ccc(C(=O)O)c(Cl)c2)ccc1[C@H](C)[C@](O)(c1ccc2c(c1)n(C)c(=O)n2C)C(F)(F)F

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CMA1 P23946 10/20 0.37
BRD4 O60885 1/20 0.36
BRPF1 P55201 1/20 0.36
TRIM24 O15164 1/20 0.35
S1PR2 O95136 1/20 0.34
PPARG P37231 1/20 0.32
PPARD Q03181 1/20 0.32
PPARA Q07869 1/20 0.32
ALDH1A1 P00352 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
MAPT P10636 1/20 0.32
CYP2C9 P11712 1/20 0.32
HPGD P15428 1/20 0.32
CYP2C19 P33261 1/20 0.32
KMT2A Q03164 1/20 0.32
SMN1; SMN2 Q16637 2/20 0.31
GAA P10253 1/20 0.31
PLA2G4A P47712 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL474551 0.94 BRD4 (0.38) CMA1BRD4BRPF1TRIM24S1PR2
SCHEMBL12164033 0.94 BRD4 (0.38) CMA1BRD4BRPF1TRIM24S1PR2
SCHEMBL474414 0.88 CMA1 (0.36) CMA1BRD4BRPF1TRIM24S1PR2
SCHEMBL12164036 0.88 CMA1 (0.36) CMA1BRD4BRPF1TRIM24S1PR2
SCHEMBL12164055 0.87 BRPF1 (0.35) CMA1BRD4BRPF1TRIM24S1PR2
SCHEMBL474489 0.87 BRPF1 (0.35) CMA1BRD4BRPF1TRIM24S1PR2
SCHEMBL474345 0.86 BRD4 (0.36) CMA1BRD4BRPF1TRIM24PPARG
SCHEMBL12164056 0.86 BRD4 (0.38) CMA1BRD4BRPF1TRIM24PPARG
SCHEMBL474255 0.86 BRD4 (0.38) CMA1BRD4BRPF1TRIM24PPARG
SCHEMBL12163974 0.84 CMA1 (0.36) CMA1BRD4BRPF1ALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411365-B1 2,3-DIARYL- OR HETEROARYL-SUBSTITUTED 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS HOFFMANN LA ROCHE (CH) 2014-03-19 EP disclosed