SCHEMBL15580945

SCHEMBL15580945

C=C1c2ccccc2C(=O)N1c1n[nH]c2cc(O[Si](C)(C)C(C)(C)C)ccc12

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CA12 O43570 4/20 0.35
CA1 P00915 4/20 0.35
CA9 Q16790 4/20 0.35
ALPL P05186 1/20 0.33
MAPT P10636 2/20 0.31
ALDH1A1 P00352 1/20 0.31
PREP P48147 1/20 0.31
HPGD P15428 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
SCN2A Q99250 1/20 0.31
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL627934 0.93 CA12 (0.38) CA12CA1CA9ALPLMAPT
SCHEMBL628629 0.84 CA12 (0.38) CA12CA1CA9ALPLMAPT
SCHEMBL20402739 0.77 ALPL (0.35) ALPLMAPTALDH1A1HPGDSMN1; SMN2
SCHEMBL627442 0.77 ALPL (0.49) ALPLMAPTALDH1A1HPGDSMN1; SMN2
SCHEMBL15580953 0.74 MAPT (0.32) CA12CA1CA9MAPTPREP
SCHEMBL6604988 0.71 TTK (0.37) ALPLMAPTALDH1A1HPGDSMN1; SMN2
SCHEMBL2452033 0.70 ALPL (0.43) ALPLSMN1; SMN2
SCHEMBL18180085 0.70 CA12 (0.38) CA12CA1CA9MAPTPREP
SCHEMBL628214 0.70 PDPK1 (0.50) CA12CA1CA9
SCHEMBL5255810 0.69 SCN2A (0.65) CA12CA1CA9PREPSCN2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10028934-B2 Substituted indazole derivatives active as kinase inhibitiors NERVIANO MEDICAL SCIENCES S.R.L. (IT) 2018-07-24 US disclosed
US-9597317-B2 Substituted indazole derivatives active as kinase inhibitiors NERVIANO MEDICAL SCIENCES S.R.L. (IT) 2017-03-21 US disclosed
US-20160311776-A1 SUBSTITUTED INDAZOLE DERIVATIVES ACTIVE AS KINASE INHIBITIORS NERVIANO MEDICAL SCIENCES S.R.L. (IT) 2016-10-27 US disclosed
US-20160310465-A1 SUBSTITUTED INDAZOLE DERIVATIVES ACTIVE AS KINASE INHIBITIORS NERVIANO MEDICAL SCIENCES S.R.L. (IT) 2016-10-27 US disclosed
US-9408850-B2 Substituted indazole derivatives active as kinase inhibitors NERVIANO MEDICAL SCIENCES S.R.L. (IT) 2016-08-09 US disclosed
US-20140080807-A1 SUBSTITUTED INDAZOLE DERIVATIVES ACTIVE AS KINASE INHIBITORS NERVIANO MEDICAL SCIENCES S.R.L. (IT) 2014-03-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140080807-A1 SUBSTITUTED INDAZOLE DERIVATIVES ACTIVE AS KINASE INHIBITORS MAP3K1, MAP3K20, MAP3K19 CA12 4803/4885CA1 4593/4885CA9 3640/4885
US-20160310465-A1 SUBSTITUTED INDAZOLE DERIVATIVES ACTIVE AS KINASE INHIBITIORS MAP3K20, MAP3K1, MAP3K5 CA12 4799/4885CA1 4525/4885CA9 3848/4885
US-10028934-B2 Substituted indazole derivatives active as kinase inhibitiors MAP3K20, MAP3K1, MAP3K5 CA12 4799/4885CA1 4525/4885CA9 3848/4885
US-20160311776-A1 SUBSTITUTED INDAZOLE DERIVATIVES ACTIVE AS KINASE INHIBITIORS MAP3K20, MAP3K1, MAP3K5 CA12 4799/4885CA1 4525/4885CA9 3848/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.