SCHEMBL1560169

SCHEMBL1560169

NC(c1cnc2cc(Cl)ccc2n1)[C@@H]1CCNC1

nearest known ligand 0.38

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 12/20 0.38
SLC6A2 P23975 11/20 0.38
SLC6A3 Q01959 11/20 0.38
HRH4 Q9H3N8 2/20 0.37
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
CYP2D6 P10635 4/20 0.36
IRAK4 Q9NWZ3 2/20 0.36
ADORA3 P0DMS8 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1463404 0.76 HRH4 (0.40) SLC6A4SLC6A2HRH4NPC1RAB9A
SCHEMBL1558582 0.74 PIK3CG (0.43) SLC6A4SLC6A2SLC6A3NPC1RAB9A
SCHEMBL1463269 0.74 PIK3CG (0.43) SLC6A4SLC6A2SLC6A3NPC1RAB9A
SCHEMBL20023738 0.70 PDE10A (0.39) HRH4NPC1RAB9A
SCHEMBL1463401 0.68 PIK3CA (0.45) IRAK4
SCHEMBL2609314 0.67 HRH4 (0.49) HRH4NPC1RAB9AADORA3
SCHEMBL31649418 0.67 HRH4 (0.45) HRH4NPC1RAB9AADORA3
SCHEMBL4725394 0.66 PIK3CG (0.53) HRH4ADORA3
SCHEMBL30889393 0.65 FGFR3 (0.46) HRH4ADORA3
SCHEMBL5979418 0.64 SLC6A2 (0.31) SLC6A4SLC6A2SLC6A3CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2303871-A1 PYRROLIDIN-3-YLMETHYL-AMINE AS OREXIN ANTAGONISTS F. Hoffmann-La Roche AG (CH) 2011-04-06 EP disclosed
WO-2010012620-A1 PYRROLIDIN-3-YLMETHYL-AMINE AS OREXIN ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2010-02-04 WO disclosed