SCHEMBL15603268

SCHEMBL15603268

CC(C)c1ccc(-c2cn3nc(NCCc4ccc(S(N)(=O)=O)cc4)sc3n2)cc1

nearest known ligand 0.54

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CA1 P00915 15/20 0.54
CA2 P00918 15/20 0.54
CA9 Q16790 15/20 0.54
CA12 O43570 12/20 0.54
FYN P06241 5/20 0.51
CA14 Q9ULX7 2/20 0.44
CA3 P07451 1/20 0.43
CA4 P22748 1/20 0.43
CA6 P23280 1/20 0.43
CA7 P43166 1/20 0.43
CA13 Q8N1Q1 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1943789 0.89 CA2 (0.69) CA1CA2CA9CA12FYN
SCHEMBL1944265 0.87 CA1 (0.55) CA1CA2CA9CA12FYN
SCHEMBL1946905 0.85 CA1 (0.55) CA1CA2CA9CA12FYN
SCHEMBL1945596 0.84 CA12 (0.54) CA1CA2CA9CA12FYN
SCHEMBL1944821 0.84 FYN (0.48) FYN
SCHEMBL1946953 0.83 CA1 (0.55) CA1CA2CA9CA12FYN
SCHEMBL1946745 0.83 FYN (0.69) CA1CA2CA9CA12FYN
SCHEMBL1944066 0.83 FYN (0.72) CA1CA2CA9CA12FYN
SCHEMBL1946803 0.83 FYN (0.68) CA1CA2CA9CA12FYN
SCHEMBL1649750 0.82 FYN (0.60) CA1CA2CA9CA12FYN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2307425-B1 IMIDAZOTHIADIAZOLES DERIVATIVES MERCK PATENT GMBH (DE) 2014-03-26 EP claimed
EP-2307425-B1 IMIDAZOTHIADIAZOLES DERIVATIVES MERCK PATENT GMBH (DE) 2014-03-26 EP disclosed