SCHEMBL15640643

SCHEMBL15640643

CC(C)c1csc(-c2c(Cl)cccc2Cl)n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TYK2 P29597 2/20 0.41
CCR4 P51679 1/20 0.40
L3MBTL1 Q9Y468 2/20 0.36
ALDH1A1 P00352 2/20 0.36
TDP1 Q9NUW8 1/20 0.36
SHMT1 P34896 1/20 0.35
SHMT2 P34897 1/20 0.35
PANK3 Q9H999 1/20 0.35
APLNR P35414 1/20 0.34
CYP19A1 P11511 1/20 0.33
CYP1A2 P05177 2/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
GRM1 Q13255 1/20 0.33
LMNA P02545 1/20 0.33
MAPT P10636 1/20 0.33
KMT2A Q03164 1/20 0.33
TRPM8 Q7Z2W7 1/20 0.32
HAO1 Q9UJM8 3/20 0.31
FABP4 P15090 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13996109 0.83 ALDH1A1 (0.54) TYK2CCR4L3MBTL1ALDH1A1TDP1
SCHEMBL23367842 0.79 TYK2 (0.56) TYK2CCR4APLNRCYP1A2CYP2D6
SCHEMBL15640894 0.77 PDE10A (0.47) L3MBTL1ALDH1A1TDP1CYP2C9LMNA
SCHEMBL577982 0.75 CCR4 (0.33) TYK2CCR4SHMT1SHMT2PANK3
SCHEMBL2739326 0.74 GFER (0.53) ALDH1A1CYP19A1CYP1A2CYP2D6CYP2C9
SCHEMBL62767 0.73 SREBF2 (0.50) CCR4L3MBTL1ALDH1A1CYP19A1LMNA
SCHEMBL12869429 0.70 KDM4E (0.58) L3MBTL1ALDH1A1TDP1CYP19A1CYP1A2
SCHEMBL2116011 0.70 IDH1 (0.33) TYK2CCR4SHMT1SHMT2
SCHEMBL6224135 0.70 ALDH1A1 (0.45) TYK2CCR4L3MBTL1ALDH1A1TDP1
SCHEMBL13996110 0.70 ABL1 (0.43) TYK2SHMT1SHMT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8697708-B2 Azabenzothiazole compounds, compositions and methods of use F. HOFFMANN-LA ROCHE AG (CH) 2014-04-15 US disclosed