SCHEMBL15664131

SCHEMBL15664131

Cc1csc(NC(=O)Oc2nc(C3CC3)ccc2Nc2cccnc2)n1

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 3/20 0.42
PIK3CG P48736 1/20 0.41
MAPK1 P28482 2/20 0.40
POLB P06746 1/20 0.40
TSHR P16473 1/20 0.40
HSD17B10 Q99714 1/20 0.40
PDE10A Q9Y233 7/20 0.40
KMT2A Q03164 1/20 0.39
KDM4E B2RXH2 1/20 0.39
NPC1 O15118 1/20 0.39
GAA P10253 1/20 0.39
RAB9A P51151 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15664078 0.89 GRM5 (0.43) GRM5PIK3CGMAPK1HSD17B10PDE10A
SCHEMBL15663528 0.88 GRM5 (0.48) GRM5PIK3CGMAPK1POLBTSHR
Hydrochloric Acid SCHEMBL17685486 0.79 GRM5 (0.47) GRM5PIK3CGMAPK1POLBTSHR
SCHEMBL15664037 0.79 PDE10A (0.45) HSD17B10PDE10ANPC1RAB9A
SCHEMBL2832741 0.79 GRM5 (0.44) GRM5PIK3CGMAPK1HSD17B10KMT2A
SCHEMBL15663663 0.79 PDE10A (0.45) PDE10A
SCHEMBL2824997 0.78 GRM5 (0.48) GRM5PIK3CGMAPK1POLBTSHR
Hydrochloric Acid SCHEMBL17685494 0.78 NPC1 (0.48) GRM5PIK3CGMAPK1POLBTSHR
SCHEMBL2827578 0.78 GRM5 (0.50) GRM5PIK3CGMAPK1POLBTSHR
SCHEMBL15663639 0.78 GRM5 (0.44) GRM5PIK3CGMAPK1POLBKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1858854-B1 PYRIDINE-2-CARBOXAMIDE DERIVATIVES AS MGLUR5 ANTAGONISTS HOFFMANN LA ROCHE (CH) 2014-05-07 EP claimed