SCHEMBL1568037

SCHEMBL1568037

NC(=O)c1ccnc(Cc2ccc(F)c(F)c2)c1

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
FYN P06241 1/20 0.52
VNN1 O95497 1/20 0.44
KDM5A P29375 4/20 0.43
KDM5B Q9UGL1 4/20 0.43
GPR52 Q9Y2T5 1/20 0.43
MBOAT4 Q96T53 1/20 0.42
KLKB1 P03952 7/20 0.41
MAP4K1 Q92918 7/20 0.41
KDM4C Q9H3R0 2/20 0.40
DPP4 P27487 1/20 0.40
MAOA P21397 1/20 0.39
MAOB P27338 1/20 0.39
KDM5C P41229 1/20 0.39
KDM5D Q9BY66 1/20 0.39
RPS6KB1 P23443 1/20 0.38
AKT1 P31749 1/20 0.38
GRM2 Q14416 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1569191 0.85 FYN (0.48) FYNKDM5AKDM5BMBOAT4KLKB1
SCHEMBL1569159 0.82 CHEK2 (0.47) KDM5AKDM5BMBOAT4KLKB1MAP4K1
SCHEMBL1568328 0.82 MBOAT4 (0.44) FYNKDM5AKDM5BGPR52MBOAT4
SCHEMBL582010 0.82 KDM5B (0.56) FYNVNN1KDM5AKDM5BKLKB1
SCHEMBL1569175 0.82 PARP1 (0.53) KDM5AKDM5BGPR52MBOAT4KDM4C
SCHEMBL1568231 0.79 MBOAT4 (0.49) KDM5AKDM5BMBOAT4KLKB1MAP4K1
SCHEMBL1568101 0.79 MBOAT4 (0.44) KDM5AKDM5BMBOAT4KLKB1MAP4K1
SCHEMBL1569193 0.79 BRD4 (0.55) FYNKDM5AKDM5BMBOAT4KDM4C
SCHEMBL1569156 0.79 CYP17A1 (0.55) KDM5AKDM5BMBOAT4KLKB1MAP4K1
SCHEMBL1569142 0.79 PARP1 (0.53) VNN1KDM5AKDM5BMBOAT4KLKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2307379-A2 ORGANIC COMPOUNDS Novartis AG (CH) 2011-04-13 EP claimed
EP-2307379-A2 ORGANIC COMPOUNDS Novartis AG (CH) 2011-04-13 EP disclosed