SCHEMBL15711397

SCHEMBL15711397

CCCOc1cccnc1C(=O)NCc1coc(-c2ccc(O)c(OCC3CC3)c2)n1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 3/20 0.37
HCRTR2 O43614 3/20 0.37
PDE4D Q08499 3/20 0.36
PDE4A P27815 2/20 0.36
PDE4B Q07343 2/20 0.36
PDE4C Q08493 2/20 0.36
ESR1 P03372 1/20 0.35
ESR2 Q92731 1/20 0.35
PTPN1 P18031 1/20 0.35
GRM4 Q14833 4/20 0.34
TRPV1 Q8NER1 1/20 0.34
ADORA2A P29274 2/20 0.33
ADORA3 P0DMS8 1/20 0.33
ADORA2B P29275 1/20 0.33
ADORA1 P30542 1/20 0.33
SYK P43405 1/20 0.33
MELK Q14680 1/20 0.33
FFAR4 Q5NUL3 1/20 0.33
GSK3B P49841 1/20 0.33
LCLAT1 Q6UWP7 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4416877 0.92 PDE4B (0.47) HCRTR1HCRTR2PDE4DPDE4APDE4B
SCHEMBL4273698 0.85 PDE4B (0.44) HCRTR1HCRTR2PDE4DPDE4APDE4B
SCHEMBL4271738 0.85 PDE4B (0.47) PDE4DPDE4APDE4BPDE4CADORA2A
SCHEMBL4275019 0.83 PDE4A (0.43) PDE4DPDE4APDE4BPDE4CGRM4
SCHEMBL4279514 0.81 PDE4B (0.42) PDE4DPDE4APDE4BPDE4CADORA2A
SCHEMBL4284444 0.81 PDE4B (0.43) HCRTR1HCRTR2PDE4DPDE4APDE4B
SCHEMBL4278639 0.80 PDE4B (0.48) PDE4DPDE4APDE4BPDE4CLCLAT1
SCHEMBL4285870 0.80 PDE4A (0.43) PDE4DPDE4APDE4BPDE4CADORA2A
SCHEMBL4280788 0.78 PDE4B (0.47) PDE4DPDE4APDE4BPDE4C
SCHEMBL4278905 0.78 PDE4D (0.44) PDE4DPDE4APDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1954684-B1 OXAZOLE COMPOUND AND PHARMACEUTICAL COMPOSITION OTSUKA PHARMA CO LTD (JP) 2014-05-07 EP disclosed