SCHEMBL15713263

SCHEMBL15713263

CN[C@@H](C)Cn1ncc2ccc(SC)cc21

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 8/20 0.47
HTR2C P28335 8/20 0.47
HTR2B P41595 5/20 0.47
HTR1A P08908 2/20 0.47
ADRA2A P08913 2/20 0.47
ADRA2B P18089 2/20 0.47
ADRA2C P18825 2/20 0.47
HTR1D P28221 1/20 0.47
HTR7 P34969 1/20 0.47
HTR4 Q13639 1/20 0.47
KMO O15229 6/20 0.43
SLC6A4 P31645 1/20 0.42
CHRM2 P08172 4/20 0.34
CHRM1 P11229 4/20 0.34
CHRM3 P20309 4/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17694538 0.83 KMO (0.51) HTR2AHTR2CHTR2BHTR1AADRA2A
SCHEMBL905933 0.83 HTR2A (0.68) HTR2AHTR2CHTR2BHTR1AADRA2A
SCHEMBL10199642 0.83 HTR2A (0.68) HTR2AHTR2CHTR2BHTR1AADRA2A
Fumaric Acid SCHEMBL8006854 0.74 HTR2A (0.58) HTR2AHTR2CHTR2BHTR1AADRA2A
Fumaric Acid SCHEMBL8009273 0.74 HTR2A (0.58) HTR2AHTR2CHTR2BHTR1AADRA2A
Fumaric Acid SCHEMBL8009278 0.74 HTR2A (0.58) HTR2AHTR2CHTR2BHTR1AADRA2A
Ammonia Solution, Strong SCHEMBL905935 0.74 HTR2A (0.44) HTR2AHTR2CHTR2BHTR1AADRA2A
SCHEMBL24908252 0.72 NOTUM (0.43) HTR2AHTR2CHTR2BKMO
SCHEMBL8013345 0.71 HTR2A (0.52) HTR2AHTR2CHTR2BHTR1AADRA2A
SCHEMBL906040 0.69 HTR2A (0.60) HTR2AHTR2CHTR2BHTR1AADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2727585-A1 In-vivo screening method Takeda Pharmaceutical Company Limited (JP) 2014-05-07 EP disclosed