SCHEMBL15720106

SCHEMBL15720106

COCCOCCOCCOc1cc(N)cc(F)c1

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.37
MAPT P10636 1/20 0.37
APP P05067 3/20 0.36
KDM4E B2RXH2 1/20 0.36
RECQL P46063 1/20 0.36
CYP1B1 Q16678 3/20 0.35
CYP1A1 P04798 2/20 0.35
CYP1A2 P05177 2/20 0.35
NCF1 P14598 6/20 0.34
TSHR P16473 1/20 0.34
CHEK1 O14757 1/20 0.33
SYK P43405 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17197212 0.88 KDM4E (0.41) APPKDM4ERECQLCYP1B1CYP1A1
SCHEMBL15071344 0.88 KDM4E (0.41) ALDH1A1MAPTAPPKDM4ERECQL
SCHEMBL15516657 0.83 TSHR (0.40) ALDH1A1MAPTAPPKDM4ERECQL
SCHEMBL15721091 0.83 TSHR (0.40) ALDH1A1MAPTAPPKDM4ERECQL
SCHEMBL15517115 0.83 TSHR (0.40) ALDH1A1MAPTAPPKDM4ERECQL
SCHEMBL16931587 0.83 TSHR (0.40) ALDH1A1MAPTAPPKDM4ERECQL
SCHEMBL16106194 0.83 TSHR (0.40) ALDH1A1MAPTAPPKDM4ERECQL
SCHEMBL325261 0.82 SOD1 (0.39) ALDH1A1CYP1A2SYK
SCHEMBL1521997 0.80 KDM4E (0.36) APPKDM4ERECQLCYP1B1CYP1A1
SCHEMBL15720769 0.80 MAPT (0.42) ALDH1A1MAPTAPPKDM4ERECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9732063-B2 Kinase inhibitors RESPIVERT LIMITED (GB) 2017-08-15 US disclosed
EP-2925742-B1 KINASE INHIBITORS RESPIVERT LTD (GB) 2016-10-26 EP disclosed
US-20150329523-A1 KINASE INHIBITORS OXULAR ACQUISITIONS LIMITED (GB) 2015-11-19 US disclosed
EP-2925742-A1 KINASE INHIBITORS Respivert Limited (GB) 2015-10-07 EP disclosed
WO-2014076484-A1 KINASE INHIBITORS RESPIVERT LIMITED (GB) 2014-05-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150329523-A1 KINASE INHIBITORS SYK, SRC, BTK ALDH1A1 4202/4885MAPT 3795/4885APP 3400/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.