SCHEMBL15722262

SCHEMBL15722262

CNC(C)c1ccc(N2CCCN(C)CC2)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NCF1 P14598 1/20 0.57
CHKA P35790 2/20 0.53
LMNA P02545 1/20 0.50
ALDH1A1 P00352 2/20 0.46
KDM4E B2RXH2 1/20 0.46
GAA P10253 1/20 0.46
MAPT P10636 1/20 0.46
ADRA2C P18825 1/20 0.46
GFER P55789 1/20 0.46
KMT2A Q03164 1/20 0.46
PTK2B Q14289 1/20 0.46
ESR2 Q92731 1/20 0.46
CACNA2D1 P54289 3/20 0.44
SLC6A2 P23975 1/20 0.41
F10 P00742 2/20 0.41
SIGMAR1 Q99720 1/20 0.41
HDAC3 O15379 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
HTR6 P50406 1/20 0.41
SIRT6 Q8N6T7 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15247182 0.83 CHKA (0.58) NCF1CHKALMNAALDH1A1KDM4E
SCHEMBL11990247 0.78 CHKA (0.56) NCF1CHKALMNAALDH1A1KDM4E
SCHEMBL11989517 0.78 CHKA (0.53) NCF1CHKALMNAALDH1A1KDM4E
SCHEMBL24171097 0.76 CHKA (0.54) NCF1CHKALMNAALDH1A1KDM4E
SCHEMBL19977464 0.76 ALDH1A1 (0.46) LMNAALDH1A1KDM4EMAPTADRA2C
SCHEMBL101926 0.76 ALDH1A1 (0.64) CHKALMNAALDH1A1KDM4EGAA
SCHEMBL82022 0.74 CHKA (0.64) NCF1CHKALMNAALDH1A1KDM4E
SCHEMBL3156564 0.74 NPC1 (0.49) LMNAALDH1A1GAAMAPTKMT2A
SCHEMBL14146896 0.73 MAPT (0.60) NCF1CHKALMNAALDH1A1KDM4E
SCHEMBL217159 0.73 MAPT (0.85) NCF1CHKALMNAALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2124951-B1 5-CYAN0-4- (PYRROLO[2, 3B]PYRIDINE-3-YL) -PYRIMIDINE DERIVATIVES USEFUL AS PROTEIN KINASE INHIBITORS VERTEX PHARMA (US) 2014-05-21 EP disclosed