SCHEMBL15725191

SCHEMBL15725191

Cc1cc(Nc2cc(C)nc(Sc3ccc(NC(=O)c4ccccc4Cl)cc3)n2)[nH]n1

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
AURKB Q96GD4 7/20 0.56
AURKA O14965 6/20 0.56
JAK2 O60674 2/20 0.47
JAK1 P23458 2/20 0.47
BDKRB1 P46663 1/20 0.44
GRM4 Q14833 1/20 0.43
SRC P12931 1/20 0.43
GSK3B P49841 1/20 0.43
AURKC Q9UQB9 1/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
PCTP Q9UKL6 1/20 0.42
DNMT1 P26358 1/20 0.42
LMNA P02545 1/20 0.42
TP53 P04637 1/20 0.42
MAPT P10636 1/20 0.42
SMO Q99835 3/20 0.42
NR2E3 Q9Y5X4 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1056600 0.94 AURKB (0.48) AURKBAURKAJAK2JAK1BDKRB1
SCHEMBL1052804 0.87 AURKB (0.56) AURKBAURKAJAK2JAK1SRC
SCHEMBL12102863 0.86 AURKA (0.51) AURKBAURKAJAK2JAK1GRM4
SCHEMBL13004613 0.85 AURKB (0.47) AURKBAURKAJAK2JAK1SRC
SCHEMBL13004050 0.85 AURKB (0.47) AURKBAURKAJAK2JAK1SRC
SCHEMBL13004282 0.84 PTGES (0.41) AURKBAURKAJAK2JAK1BDKRB1
SCHEMBL13004609 0.84 AURKB (0.45) AURKBAURKAJAK2JAK1SRC
SCHEMBL13299472 0.84 AURKB (0.48) AURKBAURKAJAK2JAK1SRC
SCHEMBL13004614 0.82 AURKB (0.44) AURKBAURKAJAK2JAK1SRC
SCHEMBL12931472 0.81 AURKB (0.54) AURKBAURKAJAK2JAK1SRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20140141099-A1 DRUG DISCOVERY METHODS VERTEX PHARMACEUTICALS INCORPORATED 2014-05-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140141099-A1 DRUG DISCOVERY METHODS AURKB, AURKC, AURKA AURKB 1/4885AURKA 3/4885JAK2 2547/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.