SCHEMBL15749403

SCHEMBL15749403

C=[N+]([O-])c1cnc(Cl)cc1NC(C)C(F)(F)F

nearest known ligand 0.33

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 4/20 0.33
IDH2 P48735 3/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15740626 0.86 ALDH1A1 (0.36) IDH1IDH2
SCHEMBL15740596 0.86 ALDH1A1 (0.36) IDH1IDH2
SCHEMBL15740820 0.86 ALDH1A1 (0.36) IDH1IDH2
SCHEMBL17447755 0.77 IDH1 (0.38) IDH1IDH2
SCHEMBL15749031 0.76
SCHEMBL15740528 0.76 IDH1 (0.37) IDH1IDH2
SCHEMBL15749038 0.76 IDH1 (0.37) IDH1IDH2
SCHEMBL15749099 0.76 IDH1 (0.37) IDH1IDH2
SCHEMBL15740748 0.73 IDH1 (0.37) IDH1IDH2
SCHEMBL19015419 0.72 IDH1 (0.35) IDH1IDH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014081718-A1 AMINOPYRIMIDINE COMPOUNDS AS INHIBITORS OF T790M CONTAINING EGFR MUTANTS GENENTECH, INC. (US) 2014-05-30 WO disclosed