SCHEMBL15760952

SCHEMBL15760952

CNc1nc(Cl)cc2nc[nH]c(=O)c12

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 8/20 0.43
ALDH1A1 P00352 1/20 0.40
XDH P47989 1/20 0.39
SYK P43405 4/20 0.38
CHEK1 O14757 1/20 0.36
PIM1 P11309 1/20 0.36
RPS6KA3 P51812 1/20 0.36
KCNH2 Q12809 2/20 0.35
JAK2 O60674 2/20 0.35
LYN P07948 2/20 0.35
ZAP70 P43403 2/20 0.35
AURKB Q96GD4 1/20 0.35
PDPK1 O15530 2/20 0.34
IP6K1 Q92551 1/20 0.34
MKNK1 Q9BUB5 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12962037 0.80 PARP1 (0.46) PARP1ALDH1A1CHEK1PIM1RPS6KA3
SCHEMBL15760947 0.79 PARP1 (0.38) PARP1XDHSYKCHEK1PIM1
SCHEMBL1059335 0.79 PARP1 (0.44) PARP1ALDH1A1SYKPIM1KCNH2
SCHEMBL1059900 0.79 PARP1 (0.49) PARP1ALDH1A1CHEK1PIM1RPS6KA3
SCHEMBL1083326 0.79 XDH (0.44) PARP1XDHSYKKCNH2JAK2
SCHEMBL1057202 0.76 SYK (0.45) SYKJAK2
SCHEMBL14641821 0.76 PARP1 (0.43) PARP1ALDH1A1CHEK1PIM1RPS6KA3
SCHEMBL1058535 0.74 PARP1 (0.49) PARP1JAK2ZAP70
SCHEMBL1057076 0.74 JAK1 (0.41) PARP1SYKJAK2
SCHEMBL15760946 0.74 CHEK1 (0.43) CHEK1RPS6KA3JAK2ZAP70

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20140171429-A1 BICYCLIC INHIBITORS OF ALK ABBVIE INC. (US) 2014-06-19 US disclosed
US-20140155389-A1 BICYCLIC INHIBITORS OF ALK ABBVIE INC. (US) 2014-06-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140171429-A1 BICYCLIC INHIBITORS OF ALK ALK, ACVR1, ACVR1B PARP1 271/4885ALDH1A1 161/4885XDH 1213/4885
US-20140155389-A1 BICYCLIC INHIBITORS OF ALK ALK, ABL1, BOD1L1 PARP1 260/4885ALDH1A1 140/4885XDH 603/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.