SCHEMBL15775666

SCHEMBL15775666

Nc1cccc2c(=O)[nH]c(-c3ccccc3)cc12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 14/20 1.00
TNKS O95271 4/20 0.51
TNKS2 Q9H2K2 2/20 0.51
KDM4E B2RXH2 1/20 0.47
CTSV O60911 1/20 0.47
LMNA P02545 1/20 0.47
TUBB4A P04350 1/20 0.47
TP53 P04637 1/20 0.47
TUBB P07437 1/20 0.47
CTSL P07711 1/20 0.47
TUBA3C P0DPH7 1/20 0.47
HPGD P15428 1/20 0.47
TUBA1B P68363 1/20 0.47
TUBA4A P68366 1/20 0.47
TUBB4B P68371 1/20 0.47
TUBB3 Q13509 1/20 0.47
TUBB2A Q13885 1/20 0.47
TUBB8 Q3ZCM7 1/20 0.47
TUBA3E Q6PEY2 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15791062 0.87 PARP1 (0.77) PARP1TNKSTNKS2CTSVCTSL
Bromide SCHEMBL15775305 0.86 PARP1 (0.74) PARP1TNKS
SCHEMBL15775367 0.86 PARP1 (1.00) PARP1TNKSTNKS2CTSVCTSL
SCHEMBL15791061 0.86 PARP1 (1.00) PARP1TNKSTNKS2KDM4E
Bromide SCHEMBL15775831 0.86 PARP1 (0.75) PARP1TNKSTNKS2CTSVCTSL
Hydrochloric Acid SCHEMBL15775429 0.84 PARP1 (0.97) PARP1TNKSTNKS2KDM4E
Bromide SCHEMBL15775373 0.84 PARP1 (0.73) PARP1TNKSTNKS2
Bromide SCHEMBL15775611 0.83 PARP1 (0.74) PARP1TNKSKDM4ELMNAHPGD
SCHEMBL15775405 0.82 PARP1 (1.00) PARP1TNKSTNKS2KDM4ELMNA
SCHEMBL15775979 0.82 PARP1 (0.69) PARP1TNKSTNKS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014087165-A1 TANKYRASE INHIBITORS UNIVERSITY OF BATH (GB) 2014-06-12 WO disclosed