SCHEMBL15775755

SCHEMBL15775755

Cc1cc(N2CCC(C(=O)O)CC2)c2nsnc2n1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.57
HSD17B10 Q99714 5/20 0.57
NPSR1 Q6W5P4 3/20 0.57
USP2 O75604 2/20 0.57
HPGD P15428 2/20 0.57
KMT2A Q03164 5/20 0.43
ALDH1A1 P00352 5/20 0.43
MEN1 O00255 3/20 0.43
CYP2C19 P33261 1/20 0.40
TSHR P16473 2/20 0.39
GAA P10253 2/20 0.39
CASP1 P29466 1/20 0.39
CASP7 P55210 1/20 0.39
TP53 P04637 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
TDP1 Q9NUW8 2/20 0.38
NOTUM Q6P988 1/20 0.38
NEK2 P51955 1/20 0.37
LMNA P02545 1/20 0.37
MAPT P10636 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15790595 0.86 ALDH1A1 (0.55) KDM4EHSD17B10NPSR1HPGDKMT2A
SCHEMBL15790597 0.80 KMT2A (0.48) NPSR1USP2KMT2AALDH1A1MEN1
SCHEMBL15776680 0.78 NPC1 (0.50) USP2KMT2AALDH1A1MEN1CYP2C19
SCHEMBL15775592 0.78 KDM4E (0.48) KDM4EHSD17B10NPSR1USP2HPGD
SCHEMBL15790592 0.76 MAPT (0.51) KMT2AMEN1TSHRTP53LMNA
SCHEMBL5844330 0.73 KDM4E (1.00) KDM4EHSD17B10NPSR1USP2HPGD
SCHEMBL15775983 0.72 NEK2 (0.49) KDM4EHSD17B10NPSR1USP2HPGD
SCHEMBL16695435 0.68 NOTUM (0.65) KDM4EHSD17B10NPSR1USP2HPGD
SCHEMBL13494044 0.68 KDM4E (0.81) KDM4EHSD17B10NPSR1USP2HPGD
SCHEMBL3256156 0.68 KDM4E (0.62) KDM4EHSD17B10NPSR1USP2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014086453-A1 AZAHETEROBICYCLIC COMPOUNDS MERCK PATENT GMBH (DE) 2014-06-12 WO claimed
WO-2014086453-A1 AZAHETEROBICYCLIC COMPOUNDS MERCK PATENT GMBH (DE) 2014-06-12 WO disclosed