SCHEMBL1582470

SCHEMBL1582470

O=C(c1ccc(F)cc1)C1CCN(CCc2ccccc2)CC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 7/20 0.87
HTR2C P28335 4/20 0.87
HTR7 P34969 4/20 0.87
HTR6 P50406 4/20 0.87
KDM4E B2RXH2 1/20 0.84
CYP1A2 P05177 1/20 0.84
CYP3A4 P08684 1/20 0.84
CYP2D6 P10635 1/20 0.84

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7418228 0.99 HTR2A (0.85) HTR2AHTR2CHTR7HTR6KDM4E
SCHEMBL4211202 0.91 HTR2A (1.00) HTR2AHTR2CHTR7HTR6KDM4E
SCHEMBL7839803 0.90 HTR2A (1.00) HTR2AHTR2CHTR7HTR6KDM4E
Hydrochloric Acid SCHEMBL9375390 0.90 HTR2A (0.98) HTR2AHTR2CHTR7HTR6KDM4E
SCHEMBL9373922 0.90 HTR2A (0.98) HTR2AHTR2CHTR7HTR6KDM4E
Hydrochloric Acid SCHEMBL9374754 0.89 HTR2A (0.95) HTR2AHTR2CHTR7HTR6KDM4E
Oxalic Acid SCHEMBL467239 0.89 HTR2A (0.95) HTR2AHTR2CHTR7HTR6KDM4E
Hydrochloric Acid SCHEMBL7828801 0.89 HTR2A (0.97) HTR2AHTR2CHTR7HTR6KDM4E
SCHEMBL1583307 0.87 HTR2A (0.88) HTR2AHTR2CHTR7HTR6KDM4E
SCHEMBL9172271 0.87 HTR2A (0.82) HTR2AHTR2CHTR7HTR6KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546100-B1 NEW BENZOYL PIPERIDINE COMPOUNDS SK HOLDINGS CO LTD (KR) 2011-04-20 EP claimed
EP-0229391-B1 PIPERIDINE DERIVATE, ITS USE AND PHARMACEUTICAL COMPOSITION CONTAINING IT Eisai Co., Ltd. (JP) 1992-07-29 EP claimed
WO-2004018423-A1 NEW BENZOYL PIPERIDINE COMPOUNDS SK CORPORATION (KR) 2004-03-04 WO disclosed
EP-0360275-B1 Imidazole antiarrhythmics MERRELL DOW PHARMA (US) 1994-01-12 EP disclosed
US-5198449-A N-substituted alpha-arylazacycloalkylmethanamines and their use as cardiovascular agents A. H. ROBINS COMPANY INCORPORATED (US) 1993-03-30 US disclosed
EP-0360275-A2 Imidazole antiarrhythmics MERRELL DOW PHARMACEUTICALS INC. (US) 1990-03-28 EP disclosed
US-4868194-A Imidazole antiarrhythmics MERRELL DOW PHARMACEUTICALS INC. (US) 1989-09-19 US disclosed