SCHEMBL9373922

SCHEMBL9373922

O=C(c1ccc(F)cc1)C1CCN(CCCCCc2ccccc2)CC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 5/20 0.98
KDM4E B2RXH2 1/20 0.98
CYP1A2 P05177 1/20 0.98
CYP3A4 P08684 1/20 0.98
CYP2D6 P10635 1/20 0.98
HTR2C P28335 3/20 0.71
HTR7 P34969 3/20 0.71
HTR6 P50406 3/20 0.71
KCNH2 Q12809 2/20 0.71

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9374754 0.99 HTR2A (0.95) HTR2AKDM4ECYP1A2CYP3A4CYP2D6
SCHEMBL4211202 0.99 HTR2A (1.00) HTR2AKDM4ECYP1A2CYP3A4CYP2D6
Hydrochloric Acid SCHEMBL9375390 0.98 HTR2A (0.98) HTR2AKDM4ECYP1A2CYP3A4CYP2D6
Oxalic Acid SCHEMBL467239 0.96 HTR2A (0.95) HTR2AKDM4ECYP1A2CYP3A4CYP2D6
SCHEMBL1582470 0.90 HTR2A (0.87) HTR2AKDM4ECYP1A2CYP3A4CYP2D6
SCHEMBL7368435 0.90 HTR2A (0.83) HTR2AKDM4ECYP1A2CYP3A4CYP2D6
Hydrochloric Acid SCHEMBL7418228 0.89 HTR2A (0.85) HTR2AKDM4ECYP1A2CYP3A4CYP2D6
SCHEMBL7252912 0.86 HTR2A (0.77) HTR2AKDM4ECYP1A2CYP3A4CYP2D6
Hydrochloric Acid SCHEMBL9650868 0.85 HTR2A (0.82) HTR2AKDM4ECYP1A2CYP3A4CYP2D6
SCHEMBL27497536 0.83 HTR2A (0.72) HTR2AKDM4ECYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0294183-B1 Use of ethylamine derivatives as antihypertensive agents AJINOMOTO KK (JP) 1994-03-30 EP claimed
EP-0294183-A1 Use of ethylamine derivatives as antihypertensive agents AJINOMOTO CO., INC. (JP) 1988-12-07 EP claimed
EP-0294183-B1 Use of ethylamine derivatives as antihypertensive agents AJINOMOTO KK (JP) 1994-03-30 EP disclosed
US-5231105-A Ethylamine derivatives and antihypertensives containing the same AJINOMOTO CO., INC. (JP) 1993-07-27 US disclosed
EP-0294183-A1 Use of ethylamine derivatives as antihypertensive agents AJINOMOTO CO., INC. (JP) 1988-12-07 EP disclosed