SCHEMBL15827017

SCHEMBL15827017

CC(C)C1NC(=O)C2(C)CSC(=N2)C2=CCC(=N2)CNC(=O)CC(/C=C/CCS)OC1=O

nearest known ligand 0.70

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 20/20 0.70
HDAC1 Q13547 19/20 0.70
HDAC2 Q92769 18/20 0.70
HDAC6 Q9UBN7 16/20 0.70
HDAC8 Q9BY41 13/20 0.70
NCOR2 Q9Y618 8/20 0.70
HDAC10 Q969S8 5/20 0.70
HDAC11 Q96DB2 2/20 0.70
HDAC7 Q8WUI4 1/20 0.70

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL71104 1.00 HDAC3 (0.70) HDAC3HDAC1HDAC2HDAC6HDAC8
SCHEMBL12610955 0.93 HDAC3 (0.60) HDAC3HDAC1HDAC2HDAC6HDAC8
SCHEMBL15827018 0.91 HDAC3 (0.64) HDAC3HDAC1HDAC2HDAC6HDAC8
SCHEMBL18477565 0.90 HDAC3 (0.58) HDAC3HDAC1HDAC2HDAC6HDAC8
SCHEMBL15827014 0.89 HDAC3 (0.76) HDAC3HDAC1HDAC2HDAC6HDAC8
SCHEMBL18477572 0.87 HDAC3 (0.70) HDAC3HDAC1HDAC2HDAC6HDAC8
SCHEMBL19107097 0.87 HDAC3 (0.71) HDAC3HDAC1HDAC2HDAC6HDAC8
SCHEMBL12702683 0.87 HDAC3 (0.52) HDAC3HDAC1HDAC2HDAC6HDAC8
SCHEMBL15827015 0.87 HDAC3 (0.52) HDAC3HDAC1HDAC2HDAC6HDAC8
SCHEMBL18477568 0.87 HDAC3 (0.56) HDAC3HDAC1HDAC2HDAC6HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8759512-B2 Methods of preparation of macrocyclic compounds UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2014-06-24 US disclosed