SCHEMBL1584764

SCHEMBL1584764

CCC(C(CN)NCCN)[Si](C)(OC)OC

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2025596 0.84
SCHEMBL477658 0.76
SCHEMBL336402 0.74
SCHEMBL27832751 0.70
SCHEMBL17649 0.67
SCHEMBL4542054 0.66
Acetic Acid SCHEMBL15453589 0.66 CPB2 (0.32)
SCHEMBL6713980 0.66 CA12 (0.38)
SCHEMBL361861 0.64
SCHEMBL2145475 0.64

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070087025-A1 Reiteratively layered medical devices and method of preparing same FITZHUGH ANTHONY 2007-04-19 US claimed
US-20070014828-A1 Cross-linked nitric oxide-releasing polyamine coated substrates, compositions comprising same and method of making same GOVERNMENT OF THE USA, REPRESENTED BY THE SECRETARY, DEPT. OF HEALTH AND HUMAN SERVICES (US) 2007-01-18 US claimed
EP-1545798-A4 CROSS-LINKED NITRIC OXIDE-RELEASING POLYAMINE COATED SUBSTRATES, COMPOSITIONS COMPRISING SAME AND METHOD OF MAKING SAME US GOV HEALTH & HUMAN SERV (US) 2006-06-14 EP claimed
EP-1545798-A1 CROSS-LINKED NITRIC OXIDE-RELEASING POLYAMINE COATED SUBSTRATES, COMPOSITIONS COMPRISING SAME AND METHOD OF MAKING SAME THE GOVERNMENT OF THE UNITED STATES OF AMERICA, as represented by THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2005-06-29 EP claimed
WO-2004012874-A1 CROSS-LINKED NITRIC OXIDE-RELEASING POLYAMINE COATED SUBSTRATES, COMPOSITIONS COMPRISING SAME AND METHOD OF MAKING SAME THE GOVERNMENT OF THE UNITED STATES OF AMERICA, REPRESENTED BY THE SECRETARY, DEPT. OF HEALTH AND HUMAN SERVICES (US) 2004-02-12 WO claimed
US-9187501-B2 Nitric oxide-releasing nanorods and their methods of use THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 2015-11-17 US disclosed
US-20140134321-A1 NITRIC OXIDE-RELEASING COATINGS THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 2014-05-15 US disclosed
US-20140065200-A1 NITRIC OXIDE-RELEASING NANORODS AND THEIR METHODS OF USE THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 2014-03-06 US disclosed
EP-2488591-A1 NITRIC OXIDE-RELEASING COATINGS Novan, Inc. (US) 2012-08-22 EP disclosed
WO-2011047013-A1 NITRIC OXIDE-RELEASING COATINGS NOVAN, INC. (US) 2011-04-21 WO disclosed
US-20110086234-A1 NITRIC OXIDE-RELEASING COATINGS NATIONAL INSTITUTES OF HEALTH-DIRECTOR DEITR 2011-04-14 US disclosed
US-20070087025-A1 Reiteratively layered medical devices and method of preparing same FITZHUGH ANTHONY 2007-04-19 US disclosed
US-20070014828-A1 Cross-linked nitric oxide-releasing polyamine coated substrates, compositions comprising same and method of making same GOVERNMENT OF THE USA, REPRESENTED BY THE SECRETARY, DEPT. OF HEALTH AND HUMAN SERVICES (US) 2007-01-18 US disclosed
EP-1545798-A4 CROSS-LINKED NITRIC OXIDE-RELEASING POLYAMINE COATED SUBSTRATES, COMPOSITIONS COMPRISING SAME AND METHOD OF MAKING SAME US GOV HEALTH & HUMAN SERV (US) 2006-06-14 EP disclosed
EP-1545798-A1 CROSS-LINKED NITRIC OXIDE-RELEASING POLYAMINE COATED SUBSTRATES, COMPOSITIONS COMPRISING SAME AND METHOD OF MAKING SAME THE GOVERNMENT OF THE UNITED STATES OF AMERICA, as represented by THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2005-06-29 EP disclosed
WO-2004012874-A1 CROSS-LINKED NITRIC OXIDE-RELEASING POLYAMINE COATED SUBSTRATES, COMPOSITIONS COMPRISING SAME AND METHOD OF MAKING SAME THE GOVERNMENT OF THE UNITED STATES OF AMERICA, REPRESENTED BY THE SECRETARY, DEPT. OF HEALTH AND HUMAN SERVICES (US) 2004-02-12 WO disclosed