SCHEMBL15850641

SCHEMBL15850641

CN(C)Cc1ccccc1N(C)C

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 12/20 0.48
SLC6A2 P23975 10/20 0.48
SLC6A3 Q01959 9/20 0.48
ALDH1A1 P00352 3/20 0.46
TSHR P16473 2/20 0.46
LMNA P02545 1/20 0.44
HTR2A P28223 3/20 0.43
CYP2D6 P10635 3/20 0.42
KDM4E B2RXH2 2/20 0.42
CYP3A4 P08684 2/20 0.42
MEN1 O00255 1/20 0.42
CYP2C19 P33261 1/20 0.42
KMT2A Q03164 1/20 0.42
HSD17B10 Q99714 1/20 0.42
CYP1A2 P05177 2/20 0.42
KCNH2 Q12809 1/20 0.42
HPGD P15428 1/20 0.42
TAAR1 Q96RJ0 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7258749 0.82 SLC6A4 (0.46) SLC6A4SLC6A2SLC6A3ALDH1A1TSHR
SCHEMBL29729780 0.82 ALDH1A1 (0.57) SLC6A4SLC6A2SLC6A3ALDH1A1TSHR
SCHEMBL125255 0.82 ALDH1A1 (0.57) SLC6A4SLC6A2SLC6A3ALDH1A1TSHR
SCHEMBL29547081 0.81 MEN1 (0.53) ALDH1A1TSHRLMNACYP2D6MEN1
SCHEMBL29408555 0.80 AR (0.50) ALDH1A1TSHRLMNACYP2D6KDM4E
SCHEMBL3871304 0.80 AR (0.50) ALDH1A1TSHRLMNACYP2D6KDM4E
SCHEMBL8734874 0.80 SLC6A4 (0.36) SLC6A4SLC6A2SLC6A3ALDH1A1TSHR
SCHEMBL709848 0.78 MAPT (0.46) ALDH1A1TSHRLMNACYP2D6KDM4E
SCHEMBL27935035 0.78 MAPT (0.41) ALDH1A1TSHRLMNACYP2D6KDM4E
SCHEMBL15224082 0.77 ALDH1A1 (0.47) ALDH1A1TSHRLMNAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 31 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3041819-B1 IMPROVED PROCESS FOR THE REDUCTIVE AMINATION OF SUBSTRATES CONTAINING A SELECTED HALOGEN TAMINCO BVBA (BE) 2020-05-13 EP claimed
US-10544087-B2 Process for the reductive amination of halogen-containing substrates TAMINCO BVBA (BE) 2020-01-28 US claimed
US-10252979-B2 Process for the reductive amination and selective hydrogenation of substrates containing a selected halogen TAMINCO BVBA (BE) 2019-04-09 US claimed
US-20170342019-A1 PROCESS FOR THE REDUCTIVE AMINATION AND SELECTIVE HYDROGENATION OF SUBSTRATES CONTAINING A SELECTED HALOGEN TAMINCO BVBA (BE) 2017-11-30 US claimed
US-20170129847-A1 PROCESS FOR THE REDUCTIVE AMINATION OF HALOGEN-CONTAINING SUBSTRATES TAMINCO BVBA (BE) 2017-05-11 US claimed
US-20160207874-A1 IMPROVED PROCESS FOR THE REDUCTIVE AMINATION AND SELECTIVE HYDROGENATION OF SUBSTRATES CONTAINING A SELECTED HALOGEN TAMINCO BVBA (BE) 2016-07-21 US claimed
EP-3041819-A1 IMPROVED PROCESS FOR THE REDUCTIVE AMINATION AND SELECTIVE HYDROGENATION OF SUBSTRATES CONTAINING A SELECTED HALOGEN Taminco bvba (BE) 2016-07-13 EP claimed
WO-2015032653-A1 IMPROVED PROCESS FOR THE REDUCTIVE AMINATION AND SELECTIVE HYDROGENATION OF SUBSTRATES CONTAINING A SELECTED HALOGEN TAMINCO (BE) 2015-03-12 WO claimed
EP-3374344-B1 IMPROVED PROCESS FOR THE REDUCTIVE AMINATION OF HALOGEN-CONTAINING SUBSTRATES TAMINCO BV (BE) 2023-10-04 EP disclosed
EP-3041819-B1 IMPROVED PROCESS FOR THE REDUCTIVE AMINATION OF SUBSTRATES CONTAINING A SELECTED HALOGEN TAMINCO BVBA (BE) 2020-05-13 EP disclosed
CN-107001235-B Improved process for reductive amination of halogen-containing materials 塔明克有限公司 2020-05-12 CN disclosed
US-10544087-B2 Process for the reductive amination of halogen-containing substrates TAMINCO BVBA (BE) 2020-01-28 US disclosed
US-10464879-B2 Process for the reductive amination of halogen-containing substrates TAMINCO BVBA (BE) 2019-11-05 US disclosed
EP-3215480-B1 IMPROVED PROCESS FOR THE REDUCTIVE AMINATION OF HALOGEN-CONTAINING SUBSTRATES TAMINCO BVBA (BE) 2019-08-14 EP disclosed
CN-106034401-A Improved process for reductive amination and selective hydrogenation of substrates containing selected halogens 塔明克公司 2016-10-19 CN disclosed
US-20160207874-A1 IMPROVED PROCESS FOR THE REDUCTIVE AMINATION AND SELECTIVE HYDROGENATION OF SUBSTRATES CONTAINING A SELECTED HALOGEN TAMINCO BVBA (BE) 2016-07-21 US disclosed
EP-3041819-A1 IMPROVED PROCESS FOR THE REDUCTIVE AMINATION AND SELECTIVE HYDROGENATION OF SUBSTRATES CONTAINING A SELECTED HALOGEN Taminco bvba (BE) 2016-07-13 EP disclosed
WO-2016071410-A1 IMPROVED PROCESS FOR THE REDUCTIVE AMINATION OF HALOGEN-CONTAINING SUBSTRATES TAMINCO (BE) 2016-05-12 WO disclosed
WO-2015032653-A1 IMPROVED PROCESS FOR THE REDUCTIVE AMINATION AND SELECTIVE HYDROGENATION OF SUBSTRATES CONTAINING A SELECTED HALOGEN TAMINCO (BE) 2015-03-12 WO disclosed
EP-2749563-A1 Binuclear metal(I) complexes for use in optoelectronics cynora GmbH (DE) 2014-07-02 EP disclosed