SCHEMBL1585765

SCHEMBL1585765

O=C(O)CNC(=O)c1c(O)c2nc3ccccc3n2n(Cc2cccc(F)c2)c1=O

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
EGLN1 Q9GZT9 9/20 0.47
EGLN3 Q9H6Z9 5/20 0.45
HIF1A Q16665 3/20 0.44
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 1/20 0.39
ALDH1A1 P00352 1/20 0.39
GAA P10253 1/20 0.39
MAPT P10636 1/20 0.39
KMT2A Q03164 1/20 0.39
HSD17B13 Q7Z5P4 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1585687 0.91 EGLN1 (0.56) EGLN1EGLN3
SCHEMBL1586363 0.85 EGLN1 (0.50) EGLN1EGLN3HIF1AMEN1MAPT
SCHEMBL1585642 0.85 EGLN1 (0.50) EGLN1EGLN3
SCHEMBL1585836 0.85 EGLN1 (0.48) EGLN1EGLN3HIF1AMEN1ALDH1A1
SCHEMBL1585761 0.84 EGLN1 (0.53) EGLN1EGLN3
SCHEMBL1585825 0.84 EGLN1 (0.48) EGLN1EGLN3
SCHEMBL1586373 0.82 EGLN3 (0.45) EGLN1EGLN3HIF1AALDH1A1MAPT
SCHEMBL1585792 0.82 KDM4E (0.48) EGLN1EGLN3HIF1AKDM4EMEN1
SCHEMBL1586485 0.82 EGLN1 (0.47) EGLN1EGLN3HIF1A
SCHEMBL1585822 0.82 EGLN1 (0.47) EGLN1EGLN3HIF1AKDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011048611-A1 NOVEL FUSED PYRIDAZINE DERIVATIVES TORRENT PHARMACEUTICALS LIMITED (IN) 2011-04-28 WO claimed
WO-2011048611-A1 NOVEL FUSED PYRIDAZINE DERIVATIVES TORRENT PHARMACEUTICALS LIMITED (IN) 2011-04-28 WO disclosed