SCHEMBL1586464

SCHEMBL1586464

CC(c1ccccc1)N1CCC(N)(N)CC1

nearest known ligand 0.68

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.68
OPRL1 P41146 7/20 0.63
OPRM1 P35372 6/20 0.63
OPRD1 P41143 6/20 0.63
OPRK1 P41145 6/20 0.63
MC4R P32245 1/20 0.59
ALDH1A1 P00352 1/20 0.45
CHRM2 P08172 2/20 0.43
CHRM1 P11229 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1586755 0.83 CYP2D6 (0.59) CYP2D6OPRL1OPRM1OPRD1OPRK1
SCHEMBL6706135 0.82 CYP2D6 (1.00) CYP2D6OPRL1OPRM1OPRD1OPRK1
SCHEMBL16226061 0.82 CYP2D6 (1.00) CYP2D6OPRL1OPRM1OPRD1OPRK1
SCHEMBL7264542 0.82 CYP2D6 (1.00) CYP2D6OPRL1OPRM1OPRD1OPRK1
SCHEMBL1684594 0.82 CYP2D6 (0.58) CYP2D6OPRL1OPRM1OPRD1OPRK1
SCHEMBL19343455 0.78 OPRL1 (0.59) CYP2D6OPRL1OPRM1OPRD1OPRK1
SCHEMBL10639858 0.78 OPRL1 (0.63) CYP2D6OPRL1OPRM1OPRD1OPRK1
SCHEMBL23850144 0.78 CYP2D6 (0.83) CYP2D6OPRL1OPRM1OPRD1OPRK1
SCHEMBL8983562 0.78 CYP2D6 (0.83) CYP2D6OPRL1OPRM1OPRD1OPRK1
SCHEMBL31046801 0.78 CYP2D6 (0.83) CYP2D6OPRL1OPRM1OPRD1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011050325-A1 COMPOSITIONS FOR TREATMENT OF CYSTIC FIBROSIS AND OTHER CHRONIC DISEASES VERTEX PHARMACEUTICALS INCORPORATED (US) 2011-04-28 WO disclosed