SCHEMBL15864640

SCHEMBL15864640

CC(C)n1cc(-c2cncc(-c3ccc(CN4CCOCC4)c(Cl)c3)c2)nn1

nearest known ligand 0.73

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 16/20 0.73
CYP2A13 Q16696 1/20 0.45
KCNH2 Q12809 1/20 0.41
JAK2 O60674 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15864635 0.89 LRRK2 (0.73) LRRK2KCNH2JAK2
SCHEMBL15864649 0.84 LRRK2 (1.00) LRRK2
SCHEMBL15865417 0.82 LRRK2 (0.73) LRRK2
SCHEMBL15864642 0.76 LRRK2 (0.49) LRRK2CYP2A13KCNH2JAK2
SCHEMBL15865251 0.74 LRRK2 (1.00) LRRK2
SCHEMBL15865010 0.73 LRRK2 (1.00) LRRK2
SCHEMBL15870205 0.72 LRRK2 (1.00) LRRK2
SCHEMBL15864797 0.72 LRRK2 (1.00) LRRK2
SCHEMBL15865096 0.71 LRRK2 (1.00) LRRK2
SCHEMBL15864644 0.71 LRRK2 (0.46) LRRK2CYP2A13KCNH2JAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2941425-A1 AMINOPYRIDINE DERIVED COMPOUNDS AS LRRK2 INHIBITORS H. Lundbeck A/S (DK) 2015-11-11 EP disclosed
WO-2014106612-A1 AMINOPYRIDINE DERIVED COMPOUNDS AS LRRK2 INHIBITORS H. LUNDBECK A/S (DK) 2014-07-10 WO disclosed