SCHEMBL15869622

SCHEMBL15869622

CCCCC(NC(=O)CC)=C(Cc1ccc(-c2ccccc2C#N)nc1)C(=O)OC

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.39
WNT3A P56704 2/20 0.34
RORC P51449 2/20 0.33
MME P08473 1/20 0.33
BDKRB1 P46663 1/20 0.32
FAAH O00519 1/20 0.32
FFAR1 O14842 1/20 0.32
AKR1B1 P15121 1/20 0.32
ALDH1A1 P00352 2/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
GAA P10253 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
PRKDC P78527 1/20 0.32
ATM Q13315 1/20 0.32
ATR Q13535 1/20 0.32
LTB4R2 Q9NPC1 1/20 0.32
EGLN1 Q9GZT9 1/20 0.31
PARP14 Q460N5 1/20 0.31
FLT3 P36888 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15869621 1.00 TSHR (0.39) TSHRWNT3ARORCMMEBDKRB1
SCHEMBL15869687 0.92 TSHR (0.37) TSHRWNT3ARORCFAAHFFAR1
SCHEMBL9947916 0.91 TSHR (0.40) TSHRWNT3ARORCMMEFAAH
SCHEMBL9947923 0.91 TSHR (0.40) TSHRWNT3ARORCMMEFAAH
SCHEMBL9947919 0.91 TSHR (0.40) TSHRWNT3ARORCMMEFAAH
SCHEMBL15869628 0.90 TSHR (0.35) TSHRWNT3AFAAHFFAR1AKR1B1
SCHEMBL9947942 0.83 TSHR (0.38) TSHRWNT3ARORCMMEFAAH
SCHEMBL9947933 0.83 TSHR (0.38) TSHRWNT3ARORCMMEFAAH
SCHEMBL9947939 0.83 TSHR (0.38) TSHRWNT3ARORCMMEFAAH
SCHEMBL28821695 0.82 PRKDC (0.36) TSHRWNT3ARORCFAAHFFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8778954-B2 Phenylpyridine derivative and medicinal agent comprising same KOWA COMPANY, LTD. (JP) 2014-07-15 US disclosed